TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I-Sar1-Ile8]-Ang2 from human angiotensin 2 receptor type 1 receptor expressed in HEK293 cells after 1 hr by gamma counting analys...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [125I-Sar1-Ile8]-Ang2 from human angiotensin 2 receptor type 1 receptor expressed in HEK293 cells after 1 hr by gamma counting analys...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [125I-Sar1-Ile8]-Ang2 from human angiotensin 2 receptor type 1 receptor expressed in HEK293 cells after 1 hr by gamma counting analys...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataKi: 317nMAssay Description:Displacement of [125I-Sar1-Ile8]-Ang2 from human angiotensin 2 receptor type 1 receptor expressed in HEK293 cells after 1 hr by gamma counting analys...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataKi: 2.48E+4nMAssay Description:Displacement of [125I-Sar1-Ile8]-Ang2 from human angiotensin 2 receptor type 1 receptor expressed in HEK293 cells after 1 hr by gamma counting analys...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR3More data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR4More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
University of Ioannina
Curated by ChEMBL
University of Ioannina
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]-D-Tyr6-His5-GnRH from recombinant human GnRH receptor expressed in HEK293 cell membrane measured after 16 to 19 hrs by gamma c...More data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR2bMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR2bMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 0.347nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
University of Ioannina
Curated by ChEMBL
University of Ioannina
Curated by ChEMBL
Affinity DataIC50: 0.690nMAssay Description:Displacement of [125I]-D-Tyr6-His5-GnRH from recombinant human GnRH receptor expressed in HEK293 cell membrane measured after 16 to 19 hrs by gamma c...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR5More data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 0.912nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
University of Ioannina
Curated by ChEMBL
University of Ioannina
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]-D-Tyr6-His5-GnRH from recombinant human GnRH receptor expressed in HEK293 cell membrane measured after 16 to 19 hrs by gamma c...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR4More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR3More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 3.47nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 3.47nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR5More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR5More data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 5.62nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
University of Ioannina
Curated by ChEMBL
University of Ioannina
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Displacement of [125I]-D-Tyr6-His5-GnRH from recombinant human GnRH receptor expressed in HEK293 cell membrane measured after 16 to 19 hrs by gamma c...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
University of Ioannina
Curated by ChEMBL
University of Ioannina
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]-D-Tyr6-His5-GnRH from recombinant human GnRH receptor expressed in HEK293 cell membrane measured after 16 to 19 hrs by gamma c...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR5More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR2bMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR2bMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR2bMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University
Curated by ChEMBL
South Dakota State University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University
Curated by ChEMBL
South Dakota State University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]Tyr0sauvagine from human CRF1 receptor expressed in HEK293 cell membrane after 120 mins by gamma scintillation counting analysi...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 24.0nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 30.2nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Displacement of 125[I-Sar1-Ile8]ANG II from human AT1 receptor expressed in HEK293 membranes after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University
Curated by ChEMBL
South Dakota State University
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 199nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (BAU)
Curated by ChEMBL
Bahcesehir University (BAU)
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
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