Compile Data Set for Download or QSAR
Found 514 with Last Name = 'pairaudeau' and Initial = 'g'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.0316nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.0316nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.0398nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.0501nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344999(2-(2'-chloro-4'-(N-methylmethylsulfonamido)-5-(tri...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50417445(AHR-504 | CUVPOSA | GLYCOPYRROLATE)copy SMILEScopy InChI
Affinity DataIC50: 0.126nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.126nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.126nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMedDrugBank
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.158nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMedDrugBank
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50417445(AHR-504 | CUVPOSA | GLYCOPYRROLATE)copy SMILEScopy InChI
Affinity DataIC50: 0.158nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419678(CHEMBL1945036)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419668(CHEMBL1947157)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMedDrugBank
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344993(2-(2'-chloro-4'-(methylsulfonyl)-5-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344996(2-(5'-cyano-2'-fluoro-5-(trifluoromethyl)biphenyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50417445(AHR-504 | CUVPOSA | GLYCOPYRROLATE)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344995(2-(5'-cyano-2'-methyl-5-(trifluoromethyl)biphenyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50417445(AHR-504 | CUVPOSA | GLYCOPYRROLATE)copy SMILEScopy InChI
Affinity DataIC50: 0.251nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMedDrugBank
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344992(2-(2'-chloro-4'-(ethylsulfonyl)-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50423388(CHEMBL251024)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:Antagonist activity at human P2Y12 receptor assessed as ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JD4Z2QPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50026419(CHEMBL1778628)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344998(2-(2'-methyl-4'-(N-methylmethylsulfonamido)-5-(tri...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50423387(CHEMBL437204)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at human P2Y12 receptor assessed as ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JD4Z2QPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50417445(AHR-504 | CUVPOSA | GLYCOPYRROLATE)copy SMILEScopy InChI
Affinity DataIC50: 0.501nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419702(CHEMBL1945038)copy SMILEScopy InChI
Affinity DataIC50: 0.501nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419670(CHEMBL1944691)copy SMILEScopy InChI
Affinity DataIC50: 0.501nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344975((2R)-2-(2'-chloro-4'-(ethylsulfonyl)-5-(trifluorom...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344988(2-(2',5-dichloro-4'-(methylsulfonyl)biphenyl-2-ylo...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344974((R)-2-(3'-cyano-5-(trifluoromethyl)biphenyl-2-ylox...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419674(CHEMBL1945031)copy SMILEScopy InChI
Affinity DataIC50: 0.631nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419710(CHEMBL1946768)copy SMILEScopy InChI
Affinity DataIC50: 0.631nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419669(CHEMBL1944690)copy SMILEScopy InChI
Affinity DataIC50: 0.631nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419671(CHEMBL1944693)copy SMILEScopy InChI
Affinity DataIC50: 0.794nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419679(CHEMBL1945037)copy SMILEScopy InChI
Affinity DataIC50: 0.794nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419687(CHEMBL1947151)copy SMILEScopy InChI
Affinity DataIC50: 0.794nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50345003(2-(4'-(N-methylmethylsulfonamido)-5-(trifluorometh...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344991(2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Mus musculus (mouse))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344991(2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Binding affinity to mouse CRTh2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419703(CHEMBL1945042)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50417438(CHEMBL1289653)copy SMILEScopy InChI
Affinity DataIC50: 1.26nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50417438(CHEMBL1289653)copy SMILEScopy InChI
Affinity DataIC50: 1.26nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM88K4PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50345007(2-(4'-(N,N-diethylsulfamoyl)-5-(trifluoromethyl)bi...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Rattus norvegicus)
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344991(2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Binding affinity to rat CRTh2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344984(2-(2',5-dichloro-4'-(ethylsulfonyl)biphenyl-2-ylox...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419665(CHEMBL1945299)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344982((2R)-2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluorom...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344994(2-(5-chloro-3'-cyanobiphenyl-2-yloxy)acetic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50419672(CHEMBL1944694)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Displacement of radiolabeled iodocyanopindolol from recombinant beta2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5H90PubMed
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