Affinity DataKi: 0.0940nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in U2OS cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in U2OS cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 36nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cells incubated for 1 hr by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [3H]CP-55,940 from human CB1 receptor expressed in CHO cells incubated for 1 hr by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 89nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in U2OS cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in U2OS cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 160nMAssay Description:Competitive inhibition of human recombinant CYP1A1 using 7-Ethoxyresorufin as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 190nMAssay Description:Competitive inhibition of human recombinant CYP3A5 expressed in baculovirus-infected insect cells using diltiazem as substrate incubated for 15 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 203nMAssay Description:Displacement of [3H]-HU-243 from CB2 receptor (unknown origin) expressed in African green monkey Cos7 cell membranes incubated for 90 mins by radioli...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 300nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 590nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 690nMAssay Description:Mixed type inhibition of human recombinant CYP2B6 expressed in baculovirus-infected insect cells using coumarin as substrate preincubated for 5 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Mixed type inhibition of human recombinant CYP2C19 using (S)-mephenytoin as substrate preincubated for 5 mins followed by NADPH-generating system add...More data for this Ligand-Target Pair
Affinity DataKi: 842nMAssay Description:Displacement of [3H]-HU-243 from CB1 receptor in Sabra rat brain synaptosomes incubated for 90 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Competitive inhibition of human recombinant CYP3A4 expressed in baculovirus-infected insect cells using diltiazem as substrate incubated for 15 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of 5-HT2C (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.11E+3nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in U2OS cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.11E+3nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in U2OS cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of mu-type opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.59E+3nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in U2OS cells by radioligand binding assayMore data for this Ligand-Target Pair