Affinity DataKi: 0.0130nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0240nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0890nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.214nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.226nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.244nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.354nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Inhibition of human active TRKA assessed as decrease in substrate phosphorylation incubated for 2 hrs using CSKtide as substrate in presence of ATP m...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of human TRKA at active state by kinetic based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.529nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.823nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human TRKA at inactive state by kinetic based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.83nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity against Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of human inactive TRKA assessed as decrease in substrate phosphorylation incubated for 2 hrs using CSKtide as substrate in presence of ATP...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 4.46nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 9.46nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 12.8nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 15.7nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibition of human inactive TRKA assessed as decrease in substrate phosphorylation incubated for 2 hrs using CSKtide as substrate in presence of ATP...More data for this Ligand-Target Pair
Affinity DataKi: 21.5nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity against Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 40.8nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 41.5nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 49.7nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 65.7nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Inhibition of human TRKA at inactive state by kinetic based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Inhibition of human active TRKA assessed as decrease in substrate phosphorylation incubated for 2 hrs using CSKtide as substrate in presence of ATP m...More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Binding affinity against Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 78.4nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 89.8nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Binding affinity against Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 122nMAssay Description:Binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 197nMAssay Description:Binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity against Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:Binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 876nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of human TRKA at active state by kinetic based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Binding affinity against Opioid receptor delta 1More data for this Ligand-Target Pair