Compile Data Set for Download or QSAR
Found 35 with Last Name = 'gamber' and Initial = 'gg'
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337697((R)-N-(1-cyanoethyl)-3-(5-(4-((isopropylamino)meth...)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337694((R)-N-(1-cyanoethyl)-3-(5-(4-((tetrahydro-2H-pyran...)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337698((R)-N-(1-cyanoethyl)-3-(5-(4-((isopropylamino)meth...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337694((R)-N-(1-cyanoethyl)-3-(5-(4-((tetrahydro-2H-pyran...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of human PKD3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337718(CHEMBL1683438 | N-(cyanomethyl)-3-(5-(4-((tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337694((R)-N-(1-cyanoethyl)-3-(5-(4-((tetrahydro-2H-pyran...)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of human PKD2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337719(CHEMBL1683439 | N-(2-cyanopropan-2-yl)-3-(5-(4-((t...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337696((R)-N-(1-cyanoethyl)-3-(5-(4-(4-methylpiperazin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337695(3-(5-(3-bromo-4-(4-methylpiperazin-1-yl)phenyl)-1H...)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337720((S)-N-(1-cyanoethyl)-3-(5-(4-((tetrahydro-2H-pyran...)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337713(CHEMBL1683433 | N-isopropyl-3-(5-(4-((isopropylami...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337705(CHEMBL1683423 | N-(cyanomethyl)-3-(5-(4-(4-methylp...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337711(CHEMBL1683430 | N-(cyanomethyl)-3-(5-(4-(4-methylp...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337704(CHEMBL1683422 | N-isopropyl-3-(5-(4-(4-methylpiper...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337717(CHEMBL1683437 | N-isopropyl-3-(5-(4-((tetrahydro-2...)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337702(3-(5-(3-bromo-4-(4-methylpiperazin-1-yl)phenyl)-1H...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337715(3-(5-(4-((cyclopropylamino)methyl)phenyl)-1H-pyraz...)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337714(CHEMBL1683311 | N-isopropyl-3-(5-(4-((2-methoxyeth...)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337712((S)-N-(1-cyanoethyl)-3-(5-(4-(4-methylpiperazin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337706(CHEMBL1683425 | N-(2-cyanoethyl)-3-(5-(4-(4-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337703(CHEMBL1683315 | N-isopropyl-3-(5-(6-(4-methylpiper...)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337701(CHEMBL1683313 | N-isopropyl-3-(5-(4-(4-methylpiper...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337710(3-(5-(4-(4-methylpiperazin-1-yl)phenyl)-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337708(CHEMBL1683427 | N-(2-hydroxyethyl)-3-(5-(4-(4-meth...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337709(CHEMBL1683428 | N-(2-(dimethylamino)ethyl)-3-(5-(4...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337699(CHEMBL1683442 | N-(3-(5-(4-(4-methylpiperazin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337700(3-(5-(4-(4-methylpiperazin-1-yl)phenyl)-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337716(CHEMBL1683434 | N-isopropyl-3-(5-(4-((2,2,2-triflu...)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337707(CHEMBL1683426 | N-(2-methoxyethyl)-3-(5-(4-(4-meth...)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetCalcium/calmodulin-dependent protein kinase type II subunit delta(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337694((R)-N-(1-cyanoethyl)-3-(5-(4-((tetrahydro-2H-pyran...)copy SMILEScopy InChI
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetPkd1(Rattus norvegicus)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337695(3-(5-(3-bromo-4-(4-methylpiperazin-1-yl)phenyl)-1H...)copy SMILEScopy InChI
Affinity DataEC50:  680nMAssay Description:Inhibition of PKD1 in rat neonatal ventricular myocytes expressing GFP-HDAC5 assessed as inhibition of phosphorylation-dependent HDAC5 nuclear exportMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetPkd1(Rattus norvegicus)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337696((R)-N-(1-cyanoethyl)-3-(5-(4-(4-methylpiperazin-1-...)copy SMILEScopy InChI
Affinity DataEC50:  570nMAssay Description:Inhibition of PKD1 in rat neonatal ventricular myocytes expressing GFP-HDAC5 assessed as inhibition of phosphorylation-dependent HDAC5 nuclear exportMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetPkd1(Rattus norvegicus)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337697((R)-N-(1-cyanoethyl)-3-(5-(4-((isopropylamino)meth...)copy SMILEScopy InChI
Affinity DataEC50:  530nMAssay Description:Inhibition of PKD1 in rat neonatal ventricular myocytes expressing GFP-HDAC5 assessed as inhibition of phosphorylation-dependent HDAC5 nuclear exportMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetPkd1(Rattus norvegicus)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337694((R)-N-(1-cyanoethyl)-3-(5-(4-((tetrahydro-2H-pyran...)copy SMILEScopy InChI
Affinity DataEC50:  240nMAssay Description:Inhibition of PKD1 in rat neonatal ventricular myocytes expressing GFP-HDAC5 assessed as inhibition of phosphorylation-dependent HDAC5 nuclear exportMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed
TargetPkd1(Rattus norvegicus)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50337698((R)-N-(1-cyanoethyl)-3-(5-(4-((isopropylamino)meth...)copy SMILEScopy InChI
Affinity DataEC50:  460nMAssay Description:Inhibition of PKD1 in rat neonatal ventricular myocytes expressing GFP-HDAC5 assessed as inhibition of phosphorylation-dependent HDAC5 nuclear exportMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM29WXPubMed