TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Inhibition of human PC1/3 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of human PC1/3 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of human PC1/3 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of human PC1/3 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 67nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Inhibition of human PC1/3 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 142nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 173nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 238nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 285nMAssay Description:Inhibition of recombinant human furin expressed in CHO cells using pyroGlu- Arg-Thr-Lys-Arg-AMC as the substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 312nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair