Compile Data Set for Download or QSAR
Found 41 with Last Name = 'zaman' and Initial = 'gz'
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14029((R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXA...)copy SMILEScopy InChI
Affinity DataKi:  25.1nMAssay Description:Inhibition of ROCK-1More data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14031(5-(1,4-diazepane-1-sulfonyl)-1,2-dihydroisoquinoli...)copy SMILEScopy InChI
Affinity DataKi:  31.6nMAssay Description:Inhibition of ROCK-1More data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417674(CHEMBL1643361)copy SMILEScopy InChI
Affinity DataKi:  63.1nMAssay Description:Inhibition of ROCK-1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14027(5-(1,4-diazepan-1-ylsulfonyl)isoquinoline | 5-(1,4...)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Inhibition of ROCK-1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417667(CHEMBL1643574)copy SMILEScopy InChI
Affinity DataKi:  794nMAssay Description:Displacement of [3H]dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417674(CHEMBL1643361)copy SMILEScopy InChI
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14031(5-(1,4-diazepane-1-sulfonyl)-1,2-dihydroisoquinoli...)copy SMILEScopy InChI
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of [3H]dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417668(CHEMBL1643368)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14027(5-(1,4-diazepan-1-ylsulfonyl)isoquinoline | 5-(1,4...)copy SMILEScopy InChI
Affinity DataKi:  2.51E+4nMAssay Description:Displacement of [3H]dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14029((R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXA...)copy SMILEScopy InChI
Affinity DataKi:  7.94E+4nMAssay Description:Displacement of [3H]dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417667(CHEMBL1643574)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417683(CHEMBL1643573)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14029((R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXA...)copy SMILEScopy InChI
Affinity DataIC50: 245nMAssay Description:Inhibition of ROCK-2 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417687(CHEMBL1643356)copy SMILEScopy InChI
Affinity DataIC50: 427nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14031(5-(1,4-diazepane-1-sulfonyl)-1,2-dihydroisoquinoli...)copy SMILEScopy InChI
Affinity DataIC50: 575nMAssay Description:Inhibition of ROCK-2 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417678(CHEMBL1643365)copy SMILEScopy InChI
Affinity DataIC50: 575nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417670(CHEMBL1643357)copy SMILEScopy InChI
Affinity DataIC50: 589nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14031(5-(1,4-diazepane-1-sulfonyl)-1,2-dihydroisoquinoli...)copy SMILEScopy InChI
Affinity DataIC50: 759nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417671(CHEMBL1643358)copy SMILEScopy InChI
Affinity DataIC50: 776nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417672(CHEMBL1643359)copy SMILEScopy InChI
Affinity DataIC50: 813nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14029((R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXA...)copy SMILEScopy InChI
Affinity DataIC50: 871nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417673(CHEMBL1643360)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417674(CHEMBL1643361)copy SMILEScopy InChI
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of ROCK-2 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417674(CHEMBL1643361)copy SMILEScopy InChI
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14027(5-(1,4-diazepan-1-ylsulfonyl)isoquinoline | 5-(1,4...)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of ROCK-2 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417675(CHEMBL1643362)copy SMILEScopy InChI
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417676(CHEMBL1643363)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417677(CHEMBL1643364)copy SMILEScopy InChI
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417681(CHEMBL1643571)copy SMILEScopy InChI
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417668(CHEMBL1643368)copy SMILEScopy InChI
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14029((R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXA...)copy SMILEScopy InChI
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of MCP1-mediated human THP cell migrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14027(5-(1,4-diazepan-1-ylsulfonyl)isoquinoline | 5-(1,4...)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417679(CHEMBL1643366)copy SMILEScopy InChI
Affinity DataIC50: 3.47E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417682(CHEMBL1643572)copy SMILEScopy InChI
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417684(CHEMBL1643575)copy SMILEScopy InChI
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417680(CHEMBL1643367)copy SMILEScopy InChI
Affinity DataIC50: 6.76E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14027(5-(1,4-diazepan-1-ylsulfonyl)isoquinoline | 5-(1,4...)copy SMILEScopy InChI
Affinity DataIC50: 6.92E+3nMAssay Description:Inhibition of MCP1-mediated human THP cell migrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM14031(5-(1,4-diazepane-1-sulfonyl)-1,2-dihydroisoquinoli...)copy SMILEScopy InChI
Affinity DataIC50: 6.92E+3nMAssay Description:Inhibition of MCP1-mediated human THP cell migrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417669(CHEMBL1643355)copy SMILEScopy InChI
Affinity DataIC50: 7.76E+3nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417674(CHEMBL1643361)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of MCP1-mediated human THP cell migrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
MSD

Curated by ChEMBL
LigandPNGBDBM50417685(CHEMBL1643576)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ROCK-1 by Immobilized metal ion affinity-based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GQKPubMed