Compile Data Set for Download or QSAR
Found 50 with Last Name = 'cassese' and Initial = 'h'
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078022(CHEMBL3417402)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078029(CHEMBL3417409)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078015(CHEMBL3417395)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078027(CHEMBL3417407)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078026(CHEMBL3417406)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078028(CHEMBL3417408)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078017(CHEMBL3417397)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078016(CHEMBL3417396)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078024(CHEMBL3417404)copy SMILEScopy InChI
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078027(CHEMBL3417407)copy SMILEScopy InChI
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078030(CHEMBL3417410)copy SMILEScopy InChI
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078019(CHEMBL3417399)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078018(CHEMBL3417398)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078030(CHEMBL3417410)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078030(CHEMBL3417410)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078015(CHEMBL3417395)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078017(CHEMBL3417397)copy SMILEScopy InChI
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078029(CHEMBL3417409)copy SMILEScopy InChI
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078018(CHEMBL3417398)copy SMILEScopy InChI
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078028(CHEMBL3417408)copy SMILEScopy InChI
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078019(CHEMBL3417399)copy SMILEScopy InChI
Affinity DataKi:  6.80E+3nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078023(CHEMBL3417403)copy SMILEScopy InChI
Affinity DataKi:  9.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078022(CHEMBL3417402)copy SMILEScopy InChI
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078018(CHEMBL3417398)copy SMILEScopy InChI
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078017(CHEMBL3417397)copy SMILEScopy InChI
Affinity DataKi:  1.29E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078016(CHEMBL3417396)copy SMILEScopy InChI
Affinity DataKi:  1.35E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078027(CHEMBL3417407)copy SMILEScopy InChI
Affinity DataKi:  1.55E+4nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078019(CHEMBL3417399)copy SMILEScopy InChI
Affinity DataKi:  1.58E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078024(CHEMBL3417404)copy SMILEScopy InChI
Affinity DataKi:  3.09E+4nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078025(CHEMBL3417405)copy SMILEScopy InChI
Affinity DataKi:  3.09E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078029(CHEMBL3417409)copy SMILEScopy InChI
Affinity DataKi:  3.39E+4nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078020(CHEMBL3417400)copy SMILEScopy InChI
Affinity DataKi:  6.31E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078021(CHEMBL3417401)copy SMILEScopy InChI
Affinity DataKi:  8.51E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078020(CHEMBL3417400)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078016(CHEMBL3417396)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078015(CHEMBL3417395)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078026(CHEMBL3417406)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078025(CHEMBL3417405)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078024(CHEMBL3417404)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078023(CHEMBL3417403)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078021(CHEMBL3417401)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-2 expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078020(CHEMBL3417400)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078021(CHEMBL3417401)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078022(CHEMBL3417402)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078023(CHEMBL3417403)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078025(CHEMBL3417405)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078028(CHEMBL3417408)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078026(CHEMBL3417406)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of FITC-BIM from recombinant human Bcl-XL expressed in Escherichia coli after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078015(CHEMBL3417395)copy SMILEScopy InChI
Affinity DataEC50:  8.20E+3nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))
Universit£ di Napoli"Federico II"

Curated by ChEMBL
LigandPNGBDBM50078022(CHEMBL3417402)copy SMILEScopy InChI
Affinity DataEC50:  700nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed