TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -51.4kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9nM ΔG°: -45.9kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 22nM ΔG°: -43.7kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
Affinity DataKi: 26nM ΔG°: -43.3kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
Affinity DataKi: 26nM ΔG°: -43.3kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
Affinity DataKi: 28nM ΔG°: -43.1kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 46nM ΔG°: -41.9kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
Affinity DataKi: 65nM ΔG°: -41.0kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 66nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
Affinity DataKi: 93nM ΔG°: -40.1kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 105nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 124nM ΔG°: -39.4kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 128nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 138nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 202nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 250nM ΔG°: -37.7kJ/molepH: 7.5 T: 2°CAssay Description:The Ki values were calculated based on an experimentally determined appropriate Kd value according to Cheng and Prusoff.More data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 259nMAssay Description:Displacement of [125I]-HEAT from COS cells membranes expressing human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 262nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in COS cells membranesMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 285nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 297nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development LLC
Curated by ChEMBL
Affinity DataKi: 331nMAssay Description:Displacement of [125I]-HEAT from COS cell membranes expressing human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
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