Compile Data Set for Download or QSAR
Found 31 with Last Name = 'nishimura' and Initial = 'h'
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50103533(CHEMBL3343947)copy SMILEScopy InChI
Affinity DataIC50: 0.0330nMAssay Description:Displacement of [3H]]nociceptin from human ORL1 receptor high affinity binding site expressed in African green monkey COS7 cells after 90 mins by top...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50103534(CHEMBL3343949)copy SMILEScopy InChI
Affinity DataIC50: 0.0590nMAssay Description:Displacement of [3H]]nociceptin from human ORL1 receptor high affinity binding site expressed in African green monkey COS7 cells after 90 mins by top...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)copy SMILEScopy InChI
Affinity DataIC50: 0.0840nMAssay Description:Binding affinity to human ORL1 receptor expressed in African green monkey COS7 cells assessed per mg protein after 90 mins by Scatchard plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50333104(CHEMBL389521 | H-FGGFTGARKSARKLANQ-NH2 | N/OFQ-NH2...)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMAssay Description:Displacement of [3H]nociceptin from recombinant ORL1 receptor expressed in COS7 cells by competitive receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9X65PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274449(CHEMBL505874 | FGGFTGARKSARKRKNQ)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50296841(CHEMBL556388 | FGGFTGARKSARKWRNQ)copy SMILEScopy InChI
Affinity DataIC50: 0.230nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50296842(CHEMBL559130 | FGGFTGARKSARKWKNQ)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50296843(CHEMBL555757 | FGGFTGARKSARKRWNQ)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50296844(CHEMBL558807 | FGGFTGARKSARKKWNQ)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274461(CHEMBL504587 | FGGFTGARKSARKWANQ)copy SMILEScopy InChI
Affinity DataIC50: 0.410nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMAssay Description:Displacement of [3H]]nociceptin from human ORL1 receptor expressed in African green monkey COS7 cells after 90 mins by topcount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50333104(CHEMBL389521 | H-FGGFTGARKSARKLANQ-NH2 | N/OFQ-NH2...)copy SMILEScopy InChI
Affinity DataIC50: 0.720nMAssay Description:Displacement of [3H]nociceptin from recombinant ORL1 receptor expressed in COS7 cells by competitive receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9X65PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50190305(Ac-RYYRIK-NH2 | CHEMBL437723)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]]nociceptin from human ORL1 receptor expressed in African green monkey COS7 cells after 90 mins by topcount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50102837(CHEMBL3343948)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]]nociceptin from human ORL1 receptor expressed in African green monkey COS7 cells after 90 mins by topcount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50103534(CHEMBL3343949)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Displacement of [3H]]nociceptin from human ORL1 receptor expressed in African green monkey COS7 cells after 90 mins by topcount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]]isoVa-RYYRIK-NH2 from human ORL1 receptor low affinity binding site expressed in African green monkey COS7 cells after 90 mins b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274468(CHEMBL510117 | FGGFTGARKSARKLWNQ)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50103533(CHEMBL3343947)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Displacement of [3H]isoVa-RYYRIK-NH2 from human ORL1 receptor expressed in African green monkey COS7 cells after 90 mins by topcount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50103533(CHEMBL3343947)copy SMILEScopy InChI
Affinity DataIC50: 8.5nMAssay Description:Displacement of [3H]]nociceptin from human ORL1 receptor expressed in African green monkey COS7 cells after 90 mins by topcount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50333104(CHEMBL389521 | H-FGGFTGARKSARKLANQ-NH2 | N/OFQ-NH2...)copy SMILEScopy InChI
Affinity DataKd:  0.0920nMAssay Description:Binding affinity to recombinant ORL1 receptor expressed in COS7 cells by saturation binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9X65PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50102836(CHEMBL3343946)copy SMILEScopy InChI
Affinity DataKd:  1.20nMAssay Description:Binding affinity to human ORL1 receptor expressed in African green monkey COS7 cells assessed per mg protein after 90 mins by Scatchard plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50333104(CHEMBL389521 | H-FGGFTGARKSARKLANQ-NH2 | N/OFQ-NH2...)copy SMILEScopy InChI
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at recombinant ORL1 receptor expressed in COS7 cells assessed as stimulation of GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9X65PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50333104(CHEMBL389521 | H-FGGFTGARKSARKLANQ-NH2 | N/OFQ-NH2...)copy SMILEScopy InChI
Affinity DataEC50:  13nMAssay Description:Agonist activity at recombinant ORL1 receptor expressed in COS7 cells assessed as stimulation of GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9X65PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274468(CHEMBL510117 | FGGFTGARKSARKLWNQ)copy SMILEScopy InChI
Affinity DataEC50:  50nMAssay Description:Agonist activity at rat ORL1 receptor expressed in african green monkey COS7 cells assessed as stimulation of [35S]GTPgammaS binding by radioligand r...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50296844(CHEMBL558807 | FGGFTGARKSARKKWNQ)copy SMILEScopy InChI
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at rat ORL1 receptor expressed in african green monkey COS7 cells assessed as stimulation of [35S]GTPgammaS binding by radioligand r...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50296843(CHEMBL555757 | FGGFTGARKSARKRWNQ)copy SMILEScopy InChI
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at rat ORL1 receptor expressed in african green monkey COS7 cells assessed as stimulation of [35S]GTPgammaS binding by radioligand r...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274461(CHEMBL504587 | FGGFTGARKSARKWANQ)copy SMILEScopy InChI
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at rat ORL1 receptor expressed in african green monkey COS7 cells assessed as stimulation of [35S]GTPgammaS binding by radioligand r...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50296842(CHEMBL559130 | FGGFTGARKSARKWKNQ)copy SMILEScopy InChI
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at rat ORL1 receptor expressed in african green monkey COS7 cells assessed as stimulation of [35S]GTPgammaS binding by radioligand r...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50296841(CHEMBL556388 | FGGFTGARKSARKWRNQ)copy SMILEScopy InChI
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at rat ORL1 receptor expressed in african green monkey COS7 cells assessed as stimulation of [35S]GTPgammaS binding by radioligand r...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed
TargetNociceptin receptor(Homo sapiens (Human))
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)copy SMILEScopy InChI
Affinity DataKd:  0.190nMAssay Description:Binding affinity to human ORL1 receptor expressed in African green monkey COS7 cells assessed per mg protein after 90 mins by Scatchard plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD42BNPubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274449(CHEMBL505874 | FGGFTGARKSARKRKNQ)copy SMILEScopy InChI
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at rat ORL1 receptor expressed in african green monkey COS7 cells assessed as stimulation of [35S]GTPgammaS binding by radioligand r...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB2435PubMed