Compile Data Set for Download or QSAR
Found 13 with Last Name = 'takikawa' and Initial = 'h'
TargetATP-binding cassette sub-family C member 3(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391002(CHEMBL2074599)copy SMILEScopy InChI
Affinity DataKi:  2.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44RCWPubMed
TargetABC-type glutathione-S-conjugate transporter(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391002(CHEMBL2074599)copy SMILEScopy InChI
Affinity DataKi:  5.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44RCWPubMed
TargetATP-binding cassette sub-family C member 3(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391003(CHEMBL493586)copy SMILEScopy InChI
Affinity DataKi:  7.70E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicles from Mrp3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44RCWPubMed
TargetATP-binding cassette sub-family C member 3(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)copy SMILEScopy InChI
Affinity DataKi:  8.38E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicles from Mrp3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44RCWPubMed
TargetATP-binding cassette sub-family C member 3(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM18050(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)copy SMILEScopy InChI
Affinity DataKi:  9.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicles from Mrp3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44RCWPubMed
TargetABC-type glutathione-S-conjugate transporter(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391003(CHEMBL493586)copy SMILEScopy InChI
Affinity DataKi:  1.05E+5nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44RCWPubMed
TargetABC-type glutathione-S-conjugate transporter(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)copy SMILEScopy InChI
Affinity DataKi:  3.37E+5nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44RCWPubMed
TargetABC-type glutathione-S-conjugate transporter(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM18050(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)copy SMILEScopy InChI
Affinity DataKi:  1.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44RCWPubMed
TargetCarboxypeptidase B(Sus scrofa)TBA
LigandPNGBDBM50577756(CHEMBL4876192)copy SMILES
Affinity DataIC50: 590nMAssay Description:Inhibition of carboxypeptidase B in porcine pancreas using hippuryl-L-Arg as substrate preincubated with substrate for 2 mins followed by enzyme addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP06NMPubMed
TargetBile salt export pump(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375575(CHEMBL270493)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake (Taurocholate: 1 uM) in canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5H4RPubMed
TargetBile salt export pump(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391001(CHEMBL2074736)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake (Taurocholate: 1 uM) in canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5H4RPubMed
TargetBile salt export pump(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375575(CHEMBL270493)copy SMILEScopy InChI
Affinity DataIC50: 6.19E+4nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake (Taurocholate: 1 uM) in membrane vesicles isolated from Bsep-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5H4RPubMed
TargetBile salt export pump(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50391001(CHEMBL2074736)copy SMILEScopy InChI
Affinity DataIC50: 6.79E+4nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake (Taurocholate: 1 uM) in membrane vesicles isolated from Bsep-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KW5H4RPubMed