Compile Data Set for Download or QSAR
Found 81 with Last Name = 'hansen' and Initial = 'hc'
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
ACADIA Pharmaceuticals A/S

Curated by ChEMBL
LigandPNGBDBM50093777(CHEMBL81377 | N-Cyclooctyl-N-{1-[3-(4-fluoro-pheno...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Compound was evaluated for its binding against 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HTTPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
ACADIA Pharmaceuticals A/S

Curated by ChEMBL
LigandPNGBDBM86525(AMI-193 | CAS_77445 | CHEMBL79834 | NSC_77445)copy SMILEScopy InChI
Affinity DataIC50: 0.316nMAssay Description:Compound was evaluated for its inverse agonist activity against 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HTTPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463896(CHEMBL4244412)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 1 hr by alpha-screen ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463896(CHEMBL4244412)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
ACADIA Pharmaceuticals A/S

Curated by ChEMBL
LigandPNGBDBM50093777(CHEMBL81377 | N-Cyclooctyl-N-{1-[3-(4-fluoro-pheno...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Compound was evaluated for its inverse agonist activity against 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HTTPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 4 hrs by alpha-screen as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetNucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))TBA
LigandPNGBDBM50571296(CHEMBL4873093)copy SMILES
Affinity DataIC50: 16nMAssay Description:Inhibition of BPTF in human HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0497KPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463896(CHEMBL4244412)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 5 mins by alpha-screen a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463896(CHEMBL4244412)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 4 hrs by alpha-screen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463896(CHEMBL4244412)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463898(CHEMBL4241469)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetNucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))TBA
LigandPNGBDBM50571296(CHEMBL4873093)copy SMILES
Affinity DataIC50: 30nMAssay Description:Inhibition of BPTF (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0497KPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM50514899(CHEMBL4461619)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of CECR2 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0497KPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463896(CHEMBL4244412)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 1 hr by alpha-screen ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
ACADIA Pharmaceuticals A/S

Curated by ChEMBL
LigandPNGBDBM50451131(AC-165043 | CHEMBL80093)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Compound was evaluated for its inverse agonist activity against 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HTTPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463900(CHEMBL4251258)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463895(CHEMBL4243172)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463899(CHEMBL4246969)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463895(CHEMBL4243172)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463900(CHEMBL4251258)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)copy SMILEScopy InChI
Affinity DataIC50: 274nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 5 mins by alpha-screen a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463900(CHEMBL4251258)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
TargetNucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))TBA
LigandPNGBDBM50514899(CHEMBL4461619)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of BPTF (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463899(CHEMBL4246969)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463899(CHEMBL4246969)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463898(CHEMBL4241469)copy SMILEScopy InChI
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463898(CHEMBL4241469)copy SMILEScopy InChI
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G6TPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
AMRI

Curated by ChEMBL
LigandPNGBDBM50094910(CHEMBL3589475)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50094913(CHEMBL3589482)copy SMILEScopy InChI
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
AMRI

Curated by ChEMBL
LigandPNGBDBM50094887(CHEMBL3589478)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
AMRI

Curated by ChEMBL
LigandPNGBDBM50094896(CHEMBL3589487)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
AMRI

Curated by ChEMBL
LigandPNGBDBM50094888(CHEMBL3589479)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50094897(CHEMBL3589469)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
AMRI

Curated by ChEMBL
LigandPNGBDBM50094908(CHEMBL3589473)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
AMRI

Curated by ChEMBL
LigandPNGBDBM50094899(CHEMBL3589471)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50094899(CHEMBL3589471)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50094898(CHEMBL3589470)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50094914(CHEMBL3589483)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
TargetNucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))TBA
LigandPNGBDBM50571298(CHEMBL4846726)copy SMILES
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant BPTF expressed in Escherichia coli BL21-Codonplus (DE3)-RIPL incubated for 30 mins by HTRF assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0497KPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50094900(CHEMBL3589472)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M67FCPubMed
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