Compile Data Set for Download or QSAR
Found 17 with Last Name = 'gerhards' and Initial = 'hj'
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019719(5-Fluoro-1-[1-(5-methyl-2,3-dihydro-benzo[1,4]diox...)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Binding affinity towards dopamine receptor D2 was determined by displacement of [3H]-spiroperidol from bovine nucleus caudate membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019721(1-[1-(6,7-Dimethyl-2,3-dihydro-benzo[1,4]dioxin-2-...)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019717(5-Chloro-1-[1-(2,3-dihydro-benzo[1,4]dioxin-2-ylme...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019726(1-[1-(7-Chloro-2,3-dihydro-benzo[1,4]dioxin-2-ylme...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Binding affinity towards dopamine receptor D2 was determined by displacement of [3H]-spiroperidol from bovine nucleus caudate membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019725(5-Methyl-1-[1-(6-methyl-2,3-dihydro-benzo[1,4]diox...)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019727(1-[1-(6,7-Dimethyl-2,3-dihydro-benzo[1,4]dioxin-2-...)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019724(5-Chloro-1-[1-(6-methyl-2,3-dihydro-benzo[1,4]diox...)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019718(5-Fluoro-1-[1-(6-fluoro-2,3-dihydro-benzo[1,4]diox...)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019728(5-Bromo-1-[1-(2,3-dihydro-benzo[1,4]dioxin-2-ylmet...)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019723(1-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-pip...)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019720(1-[1-(7-Fluoro-2,3-dihydro-benzo[1,4]dioxin-2-ylme...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019722(1-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-pip...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PR7TZJPubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Zentrale Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:In vitro antagonistic activity for Bradykinin receptor B2 by guinea pig ileal membrane receptor assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2028S70PubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Zentrale Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)copy SMILEScopy InChI
Affinity DataIC50: 5.40nMAssay Description:In vitro antagonistic activity for Bradykinin receptor B2 by guinea pig pulmonary artery assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2028S70PubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Zentrale Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50032158(CHEMBL2370243 | CPTA-D-Arg-Arg-Pro-Hyp-Gly-Thi-Ser...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:In vitro antagonistic activity for Bradykinin receptor B2 by guinea pig ileal membrane receptor assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2028S70PubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Zentrale Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50032158(CHEMBL2370243 | CPTA-D-Arg-Arg-Pro-Hyp-Gly-Thi-Ser...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:In vitro antagonistic activity for Bradykinin receptor B2 by guinea pig pulmonary artery assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2028S70PubMed