Compile Data Set for Download or QSAR
Found 433 with Last Name = 'mansell' and Initial = 'hl'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35836(pyrimidine-4-carboxamide, 118)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50176272((S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-ami...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]5HT from human 5HT2CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3M27PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294501(2-amino-6-(furan-2-yl)-N-((6-(methoxymethyl)pyridi...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35834(pyrimidine-4-carboxamide, 116)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294507(2-amino-6-(furan-2-yl)-N-(2-methylbenzyl)pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8XG5PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]5HT from human 5HT2CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3M27PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50176265((S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]5HT from human 5HT2CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3M27PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35829(pyrimidine-4-carboxamide, 111)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35833(pyrimidine-4-carboxamide, 115)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294508(2-amino-6-(furan-2-yl)-N-(3-methylbenzyl)pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294505(2-amino-N-(2-chlorobenzyl)-6-(furan-2-yl)pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35784(pyrimidine-4-carboxamide, 19 | pyrimidine-4-carbox...)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35784(pyrimidine-4-carboxamide, 19 | pyrimidine-4-carbox...)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35830(pyrimidine-4-carboxamide, 112)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35832(pyrimidine-4-carboxamide, 114)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35843(pyrimidine-4-carboxamide, 28)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50144846((S)-2-(5-Fluoro-6-methylsulfanyl-2,3-dihydro-indol...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8XG5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294510(2-amino-6-(furan-2-yl)-N-(2-methoxybenzyl)pyrimidi...)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35837(pyrimidine-4-carboxamide, 119)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294503(2-amino-N-(2-fluorobenzyl)-6-(furan-2-yl)pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294506(2-amino-N-(3-chlorobenzyl)-6-(furan-2-yl)pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35786(pyrimidine-4-carboxamide, 27)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35785(pyrimidine-4-carboxamide, 25)copy SMILEScopy InChI
Affinity DataKi:  4.30nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35785(pyrimidine-4-carboxamide, 25)copy SMILEScopy InChI
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294504(2-amino-N-(3-fluorobenzyl)-6-(furan-2-yl)pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35774(triazine-4-carboxamide, 6)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35835(pyrimidine-4-carboxamide, 117)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)copy SMILEScopy InChI
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]5HT from human 5HT2BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3M27PubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)copy SMILEScopy InChI
Affinity DataKi:  5.10nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8XG5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35839(pyrimidine-4-carboxamide, 121)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50144835((S)-1-Methyl-2-(6-methylsulfanyl-2,3-dihydro-indol...)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8XG5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35838(pyrimidine-4-carboxamide, 120)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35845(pyrimidine-4-carboxamide, 58)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294511(2-amino-6-(furan-2-yl)-N-(3-methoxybenzyl)pyrimidi...)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50144839((S)-2-(6-Ethylsulfanyl-5-fluoro-2,3-dihydro-indol-...)copy SMILEScopy InChI
Affinity DataKi:  6.40nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8XG5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35777(triazine-4-carboxamide, 9)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35841(pyrimidine-4-carboxamide, 123)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]5HT from human 5HT2CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3M27PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  6.90nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8XG5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294500(2-amino-N-((6-aminopyridin-2-yl)methyl)-6-(furan-2...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35776(triazine-4-carboxamide, 8)copy SMILEScopy InChI
Affinity DataKi:  7.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM50294502(2-amino-N-benzyl-6-(furan-2-yl)pyrimidine-4-carbox...)copy SMILEScopy InChI
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5V1MPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35840(pyrimidine-4-carboxamide, 122)copy SMILEScopy InChI
Affinity DataKi:  8.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50144842((S)-1-Methyl-2-(2,3,7,8-tetrahydro-furo[2,3-g]indo...)copy SMILEScopy InChI
Affinity DataKi:  8.70nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8XG5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35782(triazine-4-carboxamide, 14)copy SMILEScopy InChI
Affinity DataKi:  8.80nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35810(pyrimidine-4-carboxamide, 70)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50001915(1-(3-chlorophenyl)piperazine | CHEMBL478 | m-Chlor...)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8XG5PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35806(pyrimidine-4-carboxamide, 62)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis plc

Curated by ChEMBL
LigandPNGBDBM50001915(1-(3-chlorophenyl)piperazine | CHEMBL478 | m-Chlor...)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Displacement of [3H]5HT from human 5HT2CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3M27PubMed
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