Compile Data Set for Download or QSAR
Found 165 with Last Name = 'shy' and Initial = 'hs'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50225074((1S,3S,5S)-2-[(S)-2-amino-2-(3-hydroxy-adamantan-1...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMedDrugBank
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320120((2S,4S)-4-fluoro-1-(2-(2-methyl-4-oxo-4-(pyrrolidi...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279126(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-m...)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320120((2S,4S)-4-fluoro-1-(2-(2-methyl-4-oxo-4-(pyrrolidi...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279166(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-e...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279205(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-e...)copy SMILEScopy InChI
Affinity DataIC50: 12.3nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279086(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-e...)copy SMILEScopy InChI
Affinity DataIC50: 12.9nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320110((2S,4S)-4-fluoro-1-(2-(2-methyl-4-morpholino-4-oxo...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 13.2nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMedDrugBank
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320113((2S,4S)-4-fluoro-1-(2-(2-methyl-4-oxo-4-(piperidin...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320110((2S,4S)-4-fluoro-1-(2-(2-methyl-4-morpholino-4-oxo...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of DPP4 in presence of 50% rat serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279204(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-e...)copy SMILEScopy InChI
Affinity DataIC50: 14.6nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320123(CHEMBL1082996 | trans-N-(2-(3-chlorophenyl)cyclopr...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320120((2S,4S)-4-fluoro-1-(2-(2-methyl-4-oxo-4-(pyrrolidi...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320109((2S,4S)-4-fluoro-1-(2-(2-methyl-4-(4-(methylsulfon...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM11719((2S)-1-(2-{[4-(2,3-dihydro-1H-isoindol-2-yl)-2-met...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279125(2-[1-(2,4-Dichloro-phenyl)-4-methyl-5-(4-trifluoro...)copy SMILEScopy InChI
Affinity DataIC50: 15.9nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMedDrugBank
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279123(2-[5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-et...)copy SMILEScopy InChI
Affinity DataIC50: 16.3nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMedDrugBank
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320112((2S,4S)-1-(2-(4-(3,4-dihydropyridin-1(2H)-yl)-2-me...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320124(3-(2-((2S,4S)-2-cyano-4-fluoropyrrolidin-1-yl)-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320124(3-(2-((2S,4S)-2-cyano-4-fluoropyrrolidin-1-yl)-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320125(3-(2-((2S,4S)-2-cyano-4-fluoropyrrolidin-1-yl)-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320125(3-(2-((2S,4S)-2-cyano-4-fluoropyrrolidin-1-yl)-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320110((2S,4S)-4-fluoro-1-(2-(2-methyl-4-morpholino-4-oxo...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320119((2S,4S)-4-fluoro-1-(2-(4-((R)-3-hydroxypyrrolidin-...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279203(6-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-e...)copy SMILEScopy InChI
Affinity DataIC50: 22.8nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320119((2S,4S)-4-fluoro-1-(2-(4-((R)-3-hydroxypyrrolidin-...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320125(3-(2-((2S,4S)-2-cyano-4-fluoropyrrolidin-1-yl)-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of DPP4 in presence of 50% rat serumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320109((2S,4S)-4-fluoro-1-(2-(2-methyl-4-(4-(methylsulfon...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320116((2S,4S)-4-fluoro-1-(2-(4-((S)-2-(hydroxymethyl)pyr...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320111((2S,4S)-4-fluoro-1-(2-(2-methyl-4-oxo-4-(4-oxopipe...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320126(3-(2-((2S,4S)-2-cyano-4-fluoropyrrolidin-1-yl)-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320113((2S,4S)-4-fluoro-1-(2-(2-methyl-4-oxo-4-(piperidin...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320114((2S,4S)-4-fluoro-1-(2-(2-methyl-4-oxo-4-(thiazolid...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320104(3-(2-((2S,4S)-2-cyano-4-fluoropyrrolidin-1-yl)-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320119((2S,4S)-4-fluoro-1-(2-(4-((R)-3-hydroxypyrrolidin-...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320115((2S,4S)-4-fluoro-1-(2-(2-methyl-4-((R)-2-methylpyr...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279202(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-e...)copy SMILEScopy InChI
Affinity DataIC50: 32.6nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279239(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-m...)copy SMILEScopy InChI
Affinity DataIC50: 33.6nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279240(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-e...)copy SMILEScopy InChI
Affinity DataIC50: 33.8nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320117((2S,4S)-4-fluoro-1-(2-(4-((R)-3-fluoropyrrolidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279167(2-[4-Bromo-5-(4-chloro-phenyl)-1-(2,4-dichloro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 42.5nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279168(2-[5-(4-Chloro-phenyl)-4-cyclopropyl-1-(2,4-dichlo...)copy SMILEScopy InChI
Affinity DataIC50: 43.9nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of DPP4 in presence of 50% human serumMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279087(2-[5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-me...)copy SMILEScopy InChI
Affinity DataIC50: 47.4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50320118((2S,4S)-4-fluoro-1-(2-(4-((S)-3-hydroxypyrrolidin-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z953WPubMed
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