Compile Data Set for Download or QSAR
Found 129 with Last Name = 'tae' and Initial = 'hs'
LigandPNGBDBM50550633(CHEMBL4763515)copy SMILES
Affinity DataIC50: 0.200nMAssay Description:Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-curr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
LigandPNGBDBM50550634(CHEMBL4791366)copy SMILES
Affinity DataIC50: 1.20nMAssay Description:Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-curr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50117930((4-{1-[2-(6-Methyl-pyridin-2-yl)-ethyl]-piperidine...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human ERG by fluorescently labeled tracer binding methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50514668(CHEMBL4526368)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage cl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
LigandPNGBDBM50550631(CHEMBL4756657)copy SMILES
Affinity DataIC50: 2.40nMAssay Description:Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-curr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50601896(CHEMBL5203781)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB49T6PubMed
TargetNicotinic acetylcholine receptor alpha9/alpha10(RAT)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50032829(CHEMBL1836968)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Inhibition of rat alpha9alpha10 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
LigandPNGBDBM50550632(CHEMBL4787614)copy SMILES
Affinity DataIC50: 4.90nMAssay Description:Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-curr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246545(CHEMBL4065208)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetNicotinic acetylcholine receptor alpha9/alpha10(RAT)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50445326(CHEMBL3104239)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMAssay Description:Inhibition of rat alpha9alpha10 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
LigandPNGBDBM50570461(CHEMBL4847170)copy SMILES
Affinity DataIC50: 13nMAssay Description:Agonist activity at human GABAB expressed in HEK293T cells co-transfected with human CaV2.2 channel assessed as inhibition of CaV2.2-mediated Ba2+ pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WX6PubMed
LigandPNGBDBM50550638(CHEMBL4762233)copy SMILES
Affinity DataIC50: 19nMAssay Description:Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-curr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
LigandPNGBDBM50550636(CHEMBL4745449)copy SMILES
Affinity DataIC50: 19nMAssay Description:Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-curr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
LigandPNGBDBM50601896(CHEMBL5203781)copy SMILES
Affinity DataIC50: 21nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB49T6PubMed
LigandPNGBDBM50570462(CHEMBL4856595)copy SMILES
Affinity DataIC50: 21nMAssay Description:Agonist activity at human GABAB expressed in HEK293T cells co-transfected with human CaV2.2 channel assessed as inhibition of CaV2.2-mediated Ba2+ pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WX6PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50445326(CHEMBL3104239)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage cl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
LigandPNGBDBM50550639(CHEMBL4740566)copy SMILES
Affinity DataIC50: 23nMAssay Description:Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-curr...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246555(CHEMBL4086648)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetNicotinic acetylcholine receptor alpha9/alpha10(RAT)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50550631(CHEMBL4756657)copy SMILES
Affinity DataIC50: 28nMAssay Description:Inhibition of rat alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -80 mV holding potential ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246543(CHEMBL4087615)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246469(CHEMBL4102556)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50514670(CHEMBL4555265)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage cl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246489(CHEMBL4091441)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50514670(CHEMBL4555265)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Inhibition of human alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage clamp ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50266942(4,5-bis(4-chlorophenyl)-2-(2-isopropoxy-4-methoxyp...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Binding affinity to MDM2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66MPFPubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50601894(CHEMBL5196098)copy SMILES
Affinity DataIC50: 92nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB49T6PubMed
TargetNicotinic acetylcholine receptor alpha9/alpha10(RAT)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)copy SMILEScopy InChI
Affinity DataIC50: 109nMAssay Description:Inhibition of rat alpha9alpha10 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50514670(CHEMBL4555265)copy SMILEScopy InChI
Affinity DataIC50: 117nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes expressing alpha9:alpha10 mRNA injection ratio of 1:3 assessed as inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246496(CHEMBL4070113)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246486(CHEMBL4083663)copy SMILEScopy InChI
Affinity DataIC50: 148nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246542(CHEMBL4064669)copy SMILEScopy InChI
Affinity DataIC50: 155nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246471(CHEMBL4073990)copy SMILEScopy InChI
Affinity DataIC50: 181nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246441(CHEMBL4076799)copy SMILEScopy InChI
Affinity DataIC50: 201nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246556(CHEMBL4084608)copy SMILEScopy InChI
Affinity DataIC50: 219nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
LigandPNGBDBM50601894(CHEMBL5196098)copy SMILES
Affinity DataIC50: 219nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB49T6PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246511(CHEMBL4095317)copy SMILEScopy InChI
Affinity DataIC50: 231nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461915(CHEMBL4226390)copy SMILEScopy InChI
Affinity DataIC50: 249nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage cl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246449(CHEMBL4073257)copy SMILEScopy InChI
Affinity DataIC50: 256nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50601896(CHEMBL5203781)copy SMILES
Affinity DataIC50: 259nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB49T6PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50514669(CHEMBL4574008)copy SMILEScopy InChI
Affinity DataIC50: 266nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage cl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50601896(CHEMBL5203781)copy SMILES
Affinity DataIC50: 266nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB49T6PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246485(CHEMBL4091078)copy SMILEScopy InChI
Affinity DataIC50: 288nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50514668(CHEMBL4526368)copy SMILEScopy InChI
Affinity DataIC50: 354nMAssay Description:Inhibition of human alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage clamp ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89GSKPubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50550632(CHEMBL4787614)copy SMILES
Affinity DataIC50: 363nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -80 mV holding potentia...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR80MHPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea Advanced Institute of Science and Technology (KAIST)

Curated by ChEMBL
LigandPNGBDBM50246490(CHEMBL4092349)copy SMILEScopy InChI
Affinity DataIC50: 377nMAssay Description:Inhibition of human wild type ALK using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WF3PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Homo sapiens (Human))
Institute of Basic Science (IBS)

Curated by ChEMBL
LigandPNGBDBM50133328(CHEMBL3632807)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BN1PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50601895(CHEMBL5192422)copy SMILES
Affinity DataIC50: 500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB49T6PubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Homo sapiens (Human))
Institute of Basic Science (IBS)

Curated by ChEMBL
LigandPNGBDBM50133350(8-methoxy-beta-lapachone | CHEMBL2036880)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of His-tagged human MALT1 (catalytic domain-339-719 aa) by fluorescence based assay using 25 uM Ac-LRSR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BN1PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461911(CHEMBL4229033)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Inhibition of human alpha9/alpha10 G154N mutant nACHR (1:3) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889NFPubMed
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