TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1B(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 8.80nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 39.2nM ΔG°: -44.0kJ/mole EC50: 37nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 41nM ΔG°: -43.9kJ/mole EC50: 4.5nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 51nM ΔG°: -43.3kJ/molepH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 53.5nM ΔG°: -43.2kJ/mole EC50: 9.20nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 54nM ΔG°: -43.2kJ/mole EC50: 9.20nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 59.3nM ΔG°: -42.9kJ/mole EC50: 14.7nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP2(Homo sapiens)
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 63nM ΔG°: -42.8kJ/mole EC50: 54nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 67nM ΔG°: -42.6kJ/mole EC50: 28.6nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 100nM ΔG°: -41.6kJ/mole EC50: 860nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 143nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 171nM ΔG°: -40.2kJ/mole EC50: 60nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 230nM ΔG°: -39.4kJ/mole EC50: 54nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 249nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase Mip(Chlamydia pneumoniae)
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 315nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 339nM ΔG°: -38.4kJ/mole EC50: 223nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 370nM ΔG°: -38.2kJ/mole EC50: 243nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase Mip(Chlamydia pneumoniae)
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 399nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetOuter membrane protein MIP(Legionella pneumophila)
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 598nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP3(Homo sapiens (Human))
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 1.13E+3nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 1.30E+3nM ΔG°: -34.9kJ/mole EC50: 520nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 1.74E+3nM ΔG°: -34.2kJ/mole EC50: 700nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 2.14E+3nM ΔG°: -33.7kJ/mole EC50: 2.67E+3nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 2.89E+3nM ΔG°: -32.9kJ/mole EC50: 663nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 3.95E+3nM ΔG°: -32.1kJ/molepH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetOuter membrane protein MIP(Legionella pneumophila)
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Department of Translational Research in Psychiatry , Max Planck Institute of Psychiatry , 80804 Munich , Germany.
Curated by ChEMBL
Affinity DataKi: 6.59E+3nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 7.70E+3nM ΔG°: -30.4kJ/mole EC50: 980nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataEC50: 1.80E+3nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair