TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTPB using varying levels of pNPP as substrate preincubated for 15 mins followed by substrate ad...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTPB using varying levels of pNPP as substrate preincubated for 15 mins followed by substrate ad...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataKi: 2.16E+3nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTPB using varying levels of pNPP as substrate preincubated for 15 mins followed by substrate ad...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 990nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis full-length N-terminal His6-tagged PTPB expressed in Escherichia coli BL21 DE3 using pNPP as substrate after...More data for this Ligand-Target Pair
Affinity DataIC50: 1.46E+3nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.53E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
Affinity DataIC50: 4.45E+3nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 7.51E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 9.52E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
VNU University of Science (Vietnam National University
Curated by ChEMBL
VNU University of Science (Vietnam National University
Curated by ChEMBL
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 2.56E+4nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 2.82E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.25E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.32E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.51E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.53E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.53E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
VNU University of Science
Curated by ChEMBL
VNU University of Science
Curated by ChEMBL
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPB using pNPP as substrate preincubated for 15 mins followed by substrate addition and measured after 2 to...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair