Compile Data Set for Download or QSAR
Found 88 with Last Name = 'nguyen' and Initial = 'hv'
TargetCalcium/calmodulin-dependent protein kinase type 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human CAMK1A using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1G(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human CAMK1G using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human CAMK1A using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1B(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human CAMK1B using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116774(CHEMBL3608796)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116776(CHEMBL3608798)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50249319(2-(2-aminoethylamino)-4-(3-(trifluoromethyl)phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of human SYK using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human CAMK1D using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of HA-tagged CAMK1D (unknown origin) expressed in human MDA-MB-231 cells assessed as reduction in CAMK1D autophosphorylation measured afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116778(CHEMBL3608800)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of HA-tagged CAMK1D (unknown origin) expressed in human MDA-MB-231 cells assessed as reduction in CAMK1D autophosphorylation measured afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1B(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human CAMK1B using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM3263(4-Anilino quinazoline deriv. 14 | CHEMBL329672 | C...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116702(CHEMBL3608697)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116709(CHEMBL3608700)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116700(CHEMBL3608699)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545587(CHEMBL4633229 | US11530193, Example 135)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of HA-tagged CAMK1D (unknown origin) expressed in human MDA-MB-231 cells assessed as reduction in CAMK1D autophosphorylation measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116775(CHEMBL3608797)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545587(CHEMBL4633229 | US11530193, Example 135)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetDual specificity mitogen-activated protein kinase kinase 5(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human MEK5 using ERK5 as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human CAMK1D using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545586(CHEMBL4632457 | US11530193, Example 106)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545586(CHEMBL4632457 | US11530193, Example 106)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of HA-tagged CAMK1D (unknown origin) expressed in human MDA-MB-231 cells assessed as reduction in CAMK1D autophosphorylation measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116703(CHEMBL3608696)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545583(CHEMBL4644948)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116768(CHEMBL3608702)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of human MLK3 using myelin basic protein as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of human PIM1 using KKRNRTLTK as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of human BLK using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116708(CHEMBL2263368)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116773(CHEMBL3608795)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116772(CHEMBL3608794)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116704(CHEMBL3608695)copy SMILEScopy InChI
Affinity DataIC50: 67nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116771(CHEMBL3608793)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Inhibition of human SYK using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetReceptor-interacting serine/threonine-protein kinase 4(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Inhibition of human RIPK4 using histone H2A as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545584(CHEMBL4640492 | US11530193, Example 4)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545582(CHEMBL4640445 | US11530193, Example 5)copy SMILEScopy InChI
Affinity DataIC50: 101nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545585(CHEMBL4634851)copy SMILEScopy InChI
Affinity DataIC50: 115nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116781(CHEMBL2263369)copy SMILEScopy InChI
Affinity DataIC50: 155nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 168nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116770(CHEMBL3608704)copy SMILEScopy InChI
Affinity DataIC50: 173nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116705(CHEMBL460481)copy SMILEScopy InChI
Affinity DataIC50: 174nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 179nMAssay Description:Inhibition of human CAMK1D using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 186nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 5(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of human MEK5 using ERK5 as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116780(CHEMBL3608803)copy SMILEScopy InChI
Affinity DataIC50: 245nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50116777(CHEMBL3608799)copy SMILEScopy InChI
Affinity DataIC50: 254nMAssay Description:Inhibition of liver delta-5 desaturase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP552ZPubMed
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