TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Antagonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as inhibition of capsaicin-induced calcium increase after 25 ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:Antagonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as inhibition of capsaicin-induced calcium increase after 25 ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 1.34E+3nMAssay Description:Antagonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as inhibition of capsaicin-induced calcium increase after 25 ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 370nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 221nMAssay Description:Agonist activity at LPA1R (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 1.09E+3nMAssay Description:Agonist activity at LPA2 (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Agonist activity at recombinant human full-length LPA1 receptor expressed in dhfr- deficient CHO cells assessed as increase in intracellular calcium ...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 2.80E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 830nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 3.20E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 1.90E+4nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 3.20E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 2.60E+4nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 6.00E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKd: 5.60nMAssay Description:Binding affinity to LPA1 receptor (unknown origin) by cell-based backscattering interferometryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 320nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 330nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding affinity to LPA1 receptor (unknown origin) by cell-based backscattering interferometryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universit£ del Piemonte Orientale
Curated by ChEMBL
Universit£ del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Agonist activity at TRPV1 (unknown origin) expressed in human SH-SY5Y cells assessed as increase in calcium influx after 25 mins by Fluo-4 NW dye-bas...More data for this Ligand-Target Pair
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