Compile Data Set for Download or QSAR
Found 59 with Last Name = 'gomes' and Initial = 'i'
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

LigandPNGBDBM231638(SM19712)copy SMILEScopy InChI
Affinity DataIC50: 5nMpH: 5.5Assay Description:Recombinant ECE2 (32.5 ng) with a specific activity of 12 pmol/min/μg protein was generated as described previously. Secreted soluble recombinan...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6XBFPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50160900(CHEMBL181617 | N*4*-(3-Bromo-phenyl)-N*6*-(2-chlor...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 8 mins in presence of ATP by colorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XHJPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 8 mins in presence of ATP by colorimetric analysisMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50551506(CHEMBL4765122)copy SMILES
Affinity DataIC50: 504nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 8 mins in presence of ATP by colorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XHJPubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

LigandPNGBDBM231638(SM19712)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMpH: 7.4Assay Description:Recombinant ECE2 (32.5 ng) with a specific activity of 12 pmol/min/μg protein was generated as described previously. Secreted soluble recombinan...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6XBFPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50551505(CHEMBL4757104)copy SMILES
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 8 mins in presence of ATP by colorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XHJPubMed
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

LigandPNGBDBM50271179(2-(2-(quinolin-2-yl)vinyl)phenol | CHEMBL487942 | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMpH: 5.5Assay Description:Recombinant ECE2 (32.5 ng) with a specific activity of 12 pmol/min/μg protein was generated as described previously. Secreted soluble recombinan...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6XBFPubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

LigandPNGBDBM50271179(2-(2-(quinolin-2-yl)vinyl)phenol | CHEMBL487942 | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMpH: 5.5Assay Description:Recombinant ECE2 (32.5 ng) with a specific activity of 12 pmol/min/μg protein was generated as described previously. Secreted soluble recombinan...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6XBFPubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

LigandPNGBDBM50271179(2-(2-(quinolin-2-yl)vinyl)phenol | CHEMBL487942 | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMpH: 7.4Assay Description:Recombinant ECE2 (32.5 ng) with a specific activity of 12 pmol/min/μg protein was generated as described previously. Secreted soluble recombinan...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6XBFPubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

LigandPNGBDBM231638(SM19712)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMpH: 5.5Assay Description:Recombinant ECE2 (32.5 ng) with a specific activity of 12 pmol/min/μg protein was generated as described previously. Secreted soluble recombinan...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6XBFPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554767(CHEMBL4776176)copy SMILES
Affinity DataEC50:  144nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554768(CHEMBL4783765)copy SMILES
Affinity DataEC50:  85nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554769(CHEMBL4788377)copy SMILES
Affinity DataEC50:  32nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554770(CHEMBL4783653)copy SMILES
Affinity DataEC50:  163nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554771(CHEMBL4784041)copy SMILES
Affinity DataEC50:  70nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554772(CHEMBL4793926)copy SMILES
Affinity DataEC50:  264nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554773(CHEMBL4779684)copy SMILES
Affinity DataEC50:  191nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554774(CHEMBL4755700)copy SMILES
Affinity DataEC50:  380nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554775(CHEMBL4784650)copy SMILES
Affinity DataEC50:  129nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554769(CHEMBL4788377)copy SMILES
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554777(CHEMBL4751491)copy SMILES
Affinity DataEC50:  4.33E+3nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554778(CHEMBL4740220)copy SMILES
Affinity DataEC50:  1.58E+3nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)copy SMILEScopy InChI
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)copy SMILEScopy InChI
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
LigandPNGBDBM50000507((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)copy SMILEScopy InChI
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
LigandPNGBDBM50000507((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)copy SMILEScopy InChI
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
LigandPNGBDBM50554766(CHEMBL4795492)copy SMILES
Affinity DataEC50:  0.0320nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
LigandPNGBDBM50554766(CHEMBL4795492)copy SMILES
Affinity DataEC50:  0.0316nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)copy SMILEScopy InChI
Affinity DataEC50:  83nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM83396(1-(4-acetamidobenzyl)-4-phenethyl-isonipecotic aci...)copy SMILEScopy InChI
Affinity DataEC50:  945nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554762(CHEMBL4760974)copy SMILES
Affinity DataEC50:  426nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554763(CHEMBL4758061)copy SMILES
Affinity DataEC50:  2.65E+3nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554764(CHEMBL4761310)copy SMILES
Affinity DataEC50:  2.15E+3nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554766(CHEMBL4795492)copy SMILES
Affinity DataEC50:  119nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554770(CHEMBL4783653)copy SMILES
Affinity DataEC50:  605nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50000507((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554765(CHEMBL4781906)copy SMILES
Affinity DataEC50:  61nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554766(CHEMBL4795492)copy SMILES
Affinity DataEC50:  172nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554770(CHEMBL4783653)copy SMILES
Affinity DataEC50:  3.33E+3nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554774(CHEMBL4755700)copy SMILES
Affinity DataEC50:  1.02E+3nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554775(CHEMBL4784650)copy SMILES
Affinity DataEC50:  93nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554776(CHEMBL4751847)copy SMILES
Affinity DataEC50:  374nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554777(CHEMBL4751491)copy SMILES
Affinity DataEC50:  659nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554778(CHEMBL4740220)copy SMILES
Affinity DataEC50:  288nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM83396(1-(4-acetamidobenzyl)-4-phenethyl-isonipecotic aci...)copy SMILEScopy InChI
Affinity DataEC50:  812nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50000507((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)copy SMILEScopy InChI
Affinity DataEC50:  8nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554765(CHEMBL4781906)copy SMILES
Affinity DataEC50:  509nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554766(CHEMBL4795492)copy SMILES
Affinity DataEC50:  960nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554766(CHEMBL4795492)copy SMILES
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50554765(CHEMBL4781906)copy SMILES
Affinity DataEC50:  205nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1QKZPubMed
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