Compile Data Set for Download or QSAR
Found 488 with Last Name = 'lemasson' and Initial = 'i'
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357011(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356996(5-Amino-N-(4-chloro-2-fluoro-phenyl)-1-(o-tolyl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357006(5-Amino-3-ethyl-1-(3-fluoro-2-methylphenyl)-N-[5-t...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357010(5-Amino-1-(2-hydroxyphenyl)-N-(5-(trifluoromethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357002(5-Amino-3-ethyl-1-(2-methoxyphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357007(5-Amino-1-(2-fluorophenyl)-3-methyl-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356998(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357004(5-Amino-N-(5-chloro-2-pyridyl)-1-(3-fluoro-2-methy...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356997(5-Amino-N-(2-fluoro-4-(trifluoromethyl)phenyl)-1-(...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357008(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357003(5-Amino-1-(2-(2-methoxyethoxy)phenyl)-3-methyl-N-(...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356995(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357001(5-Amino-N-(5-chloropyridin-2-yl)-1-(3-fluoro-2-met...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356999((5-Amino-1-(3-fluoro-2-methylphenyl)-1H-pyrazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357000((5-Amino-1-(2-methoxyphenyl)-1H-pyrazol-4-yl)(5-ch...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357009(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(2-methoxypy...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357005(5-Amino-1-(2-ethylphenyl)-N-(5-(2,2,2-trifluoroeth...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357012(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357006(5-Amino-3-ethyl-1-(3-fluoro-2-methylphenyl)-N-[5-t...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357008(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356995(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357000((5-Amino-1-(2-methoxyphenyl)-1H-pyrazol-4-yl)(5-ch...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357004(5-Amino-N-(5-chloro-2-pyridyl)-1-(3-fluoro-2-methy...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357002(5-Amino-3-ethyl-1-(2-methoxyphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357001(5-Amino-N-(5-chloropyridin-2-yl)-1-(3-fluoro-2-met...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357007(5-Amino-1-(2-fluorophenyl)-3-methyl-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356999((5-Amino-1-(3-fluoro-2-methylphenyl)-1H-pyrazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356998(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357009(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(2-methoxypy...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356997(5-Amino-N-(2-fluoro-4-(trifluoromethyl)phenyl)-1-(...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357010(5-Amino-1-(2-hydroxyphenyl)-N-(5-(trifluoromethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356996(5-Amino-N-(4-chloro-2-fluoro-phenyl)-1-(o-tolyl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357005(5-Amino-1-(2-ethylphenyl)-N-(5-(2,2,2-trifluoroeth...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357003(5-Amino-1-(2-(2-methoxyethoxy)phenyl)-3-methyl-N-(...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357012(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Laboratoire de Chimie et de Biochimie Pharmacologiques et Toxicologiques , CNRS UMR 8601, Université Paris Descartes, Sorbonne Paris Cité , 45 rue des Saints-Pères , 75270 Paris Cedex 06 , France.

Curated by ChEMBL
LigandPNGBDBM50446782(CHEMBL3114672)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+6nMAssay Description:Antagonist activity at rat GluN1a/GluN2A receptors expressed in Xenopus laevis oocytes assessed as inhibition of L-glutamate/glucine induced current ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0BR0PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(RAT)
Laboratoire de Chimie et de Biochimie Pharmacologiques et Toxicologiques , CNRS UMR 8601, Université Paris Descartes, Sorbonne Paris Cité , 45 rue des Saints-Pères , 75270 Paris Cedex 06 , France.

Curated by ChEMBL
LigandPNGBDBM50446782(CHEMBL3114672)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+6nMAssay Description:Antagonist activity at rat GluN1a/mouse GluN2B receptors expressed in Xenopus laevis oocytes assessed as inhibition of L-glutamate/glucine induced cu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0BR0PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM82006(D-AP4 | D-APB | US9212196, L-AP4)copy SMILEScopy InChI
Affinity DataEC50:  130nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196906(US9212196, Derivative 2)copy SMILEScopy InChI
Affinity DataEC50:  110nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196907(US9212196, Derivative 3)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196908(US9212196, Derivative 4)copy SMILEScopy InChI
Affinity DataEC50:  500nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196909(US9212196, Derivative 5)copy SMILEScopy InChI
Affinity DataEC50:  280nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196910(US9212196, Derivative 6)copy SMILEScopy InChI
Affinity DataEC50:  80nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196911(US9212196, Derivative 7)copy SMILEScopy InChI
Affinity DataEC50:  130nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196912(US9212196, Derivative 8)copy SMILEScopy InChI
Affinity DataEC50:  150nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196913(US9212196, Derivative 9)copy SMILEScopy InChI
Affinity DataEC50:  380nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196914(US9212196, Derivative 10)copy SMILEScopy InChI
Affinity DataEC50:  530nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196915(US9212196, Derivative 11)copy SMILEScopy InChI
Affinity DataEC50:  480nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196916(US9212196, Derivative 12)copy SMILEScopy InChI
Affinity DataEC50:  980nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196917(US9212196, Derivative 13)copy SMILEScopy InChI
Affinity DataEC50:  1.22E+4nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
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