Compile Data Set for Download or QSAR
Found 17 with Last Name = 'mosca' and Initial = 'i'
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465610(CHEMBL4295040)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced channel currents by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465611(CHEMBL4284808)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced channel currents by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465610(CHEMBL4295040)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50133817(4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic ...)copy SMILEScopy InChI
Affinity DataIC50: 475nMAssay Description:Antagonist activity at TRPM8 (unknown origin) assessed as reduction in menthol-induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465611(CHEMBL4284808)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465615(CHEMBL4282067)copy SMILEScopy InChI
Affinity DataIC50: 865nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced channel currents by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465618(CHEMBL4291622)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465619(CHEMBL4287812)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465614(CHEMBL4292679)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465613(CHEMBL4277563)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50159505(CHEMBL1779158 | N,N-Dibenzyltryptamine)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465609(CHEMBL4277150)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465620(CHEMBL4288211)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50331290(CHEMBL1289953 | N-(3-aminopropyl)-2-(3-methylbenzy...)copy SMILEScopy InChI
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465612(CHEMBL4279001)copy SMILEScopy InChI
Affinity DataIC50: 8.20E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465616(CHEMBL4284391)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+4nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50465617(CHEMBL4280979)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced calcium flux incubated for 60 mins by Fluo-4 NW-d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN18V3PubMed