Compile Data Set for Download or QSAR
Found 148 with Last Name = 'votruba' and Initial = 'i'
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20079(5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]-1,2,3,...)copy SMILEScopy InChI
Affinity DataKi:  1.30nM ΔG°:  -52.8kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20079(5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]-1,2,3,...)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20061(5-Substituted-6-chlorouracil, 7a | 6-chloro-5-(cyc...)copy SMILEScopy InChI
Affinity DataKi:  200nM ΔG°:  -39.8kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM50310199((1-fluoro-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimid...)copy SMILEScopy InChI
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM50310200((1-hydroxy-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimi...)copy SMILEScopy InChI
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM50310201((1-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-...)copy SMILEScopy InChI
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM50310202((2-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-...)copy SMILEScopy InChI
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM50201010(((2R,3aR,4R,6R,6aR)-4-(hydroxymethyl)-6-(5-methyl-...)copy SMILEScopy InChI
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM50310203(8-(5-bromo-3-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydro...)copy SMILEScopy InChI
Affinity DataKi:  236nMAssay Description:Inhibition of human recombinant thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20069(5-Substituted-6-chlorouracil, 10e | 6-chloro-5-(th...)copy SMILEScopy InChI
Affinity DataKi:  280nM ΔG°:  -38.9kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20065(5-Substituted-6-chlorouracil, 10a | 6-chloro-5-phe...)copy SMILEScopy InChI
Affinity DataKi:  400nM ΔG°:  -38.0kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20073(5-Substituted-6-chlorouracil, 13c | 6-chloro-5-[(1...)copy SMILEScopy InChI
Affinity DataKi:  410nM ΔG°:  -37.9kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20062(5-Substituted-6-chlorouracil, 7b | 6-chloro-5-(cyc...)copy SMILEScopy InChI
Affinity DataKi:  420nM ΔG°:  -37.9kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20064(5-Substituted-6-chlorouracil, 7d | 6-chloro-5-[(2E...)copy SMILEScopy InChI
Affinity DataKi:  490nM ΔG°:  -37.5kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20075(6-Fluoro-5-phenylpyrimidine-2,4(1H,3H)-dione, 21 |...)copy SMILEScopy InChI
Affinity DataKi:  500nM ΔG°:  -37.4kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20072(5-Substituted-6-chlorouracil, 13b | 5-[(1E)-but-1-...)copy SMILEScopy InChI
Affinity DataKi:  630nM ΔG°:  -36.8kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20068(5-Substituted-6-chlorouracil, 10d | 6-chloro-5-(4-...)copy SMILEScopy InChI
Affinity DataKi:  710nM ΔG°:  -36.5kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20056(5-Substituted-6-chlorouracil, 5c | 5-butyl-6-chlor...)copy SMILEScopy InChI
Affinity DataKi:  1.03E+3nM ΔG°:  -35.5kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20059(5-Substituted-6-chlorouracil, 5f | 6-chloro-5-hept...)copy SMILEScopy InChI
Affinity DataKi:  1.06E+3nM ΔG°:  -35.5kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20071(5-Substituted-6-chlorouracil, 13a | 6-chloro-5-[(1...)copy SMILEScopy InChI
Affinity DataKi:  1.17E+3nM ΔG°:  -35.2kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20076(6-Bromo-5-phenylpyrimidine-2,4(1H,3H)-dione, 23 | ...)copy SMILEScopy InChI
Affinity DataKi:  1.21E+3nM ΔG°:  -35.1kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20066(5-Substituted-6-chlorouracil, 10b | 6-chloro-5-(3,...)copy SMILEScopy InChI
Affinity DataKi:  1.74E+3nM ΔG°:  -34.2kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20058(5-Substituted-6-chlorouracil, 5e | 6-chloro-5-hexy...)copy SMILEScopy InChI
Affinity DataKi:  1.83E+3nM ΔG°:  -34.1kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20070(5-Substituted-6-chlorouracil, 10f | 6-chloro-5-(py...)copy SMILEScopy InChI
Affinity DataKi:  3.01E+3nM ΔG°:  -32.8kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20063(5-Substituted-6-chlorouracil, 7c | 6-chloro-5-(pro...)copy SMILEScopy InChI
Affinity DataKi:  3.34E+3nM ΔG°:  -32.5kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20057(5-Substituted-6-chlorouracil, 5d | 6-chloro-5-pent...)copy SMILEScopy InChI
Affinity DataKi:  3.67E+3nM ΔG°:  -32.3kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20067(5-Substituted-6-chlorouracil, 10c | 6-chloro-5-(na...)copy SMILEScopy InChI
Affinity DataKi:  4.59E+3nM ΔG°:  -31.7kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20060(5-Substituted-6-chlorouracil, 5g | 5-benzyl-6-chlo...)copy SMILEScopy InChI
Affinity DataKi:  4.65E+3nM ΔG°:  -31.7kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20055(5-Substituted-6-chlorouracil, 5b | 6-chloro-5-prop...)copy SMILEScopy InChI
Affinity DataKi:  5.81E+3nM ΔG°:  -31.1kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20077(5-Phenyl-6-pyrrolidin-1-ylpyrimidine-2,4(1H,3H)-di...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+4nM ΔG°: >-27.9kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20078(6-[(2-Aminoethyl)amino]-5-phenylpyrimidine-2,4(1H,...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+4nM ΔG°: >-27.9kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20054(5-Substituted-6-chlorouracil, 5a | 6-chloro-5-ethy...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+4nM ΔG°: >-27.9kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Gilead Sciences Inc.

LigandPNGBDBM20074(6-Methyl-5-phenylpyrimidine-2,4(1H,3H)-dione, 16 |...)copy SMILEScopy InChI
Affinity DataKi: >2.00E+4nM ΔG°: >-27.9kJ/molepH: 6.4 T: 2°CAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043PXPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378690(CHEMBL597306)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378691(CHEMBL609919)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378689(CHEMBL599563)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378684(CHEMBL599543)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetAdenosine kinase(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50350205(CHEMBL1814774)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of human ADK using [3H]-adenosine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1CQXPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378687(CHEMBL598328)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetAdenosine kinase(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50350207(CHEMBL1814776)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human ADK expressed in Escherichia coli BL21(DE3) cells using [3H]adenosine by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50350207(CHEMBL1814776)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human ADK using [3H]-adenosine by scintillation countingMore data for this Ligand-Target Pair
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378688(CHEMBL599562)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378685(CHEMBL599544)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378692(CHEMBL611383)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378686(CHEMBL598327)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetThymidine phosphorylase(Rattus norvegicus)
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50378683(CHEMBL599132)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Inhibition of thymidine phosphorylase in T cell lymphomas of Sprague-Dawley rat in presence of 100 uM thymidine and 200 uM phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930V4KPubMed
TargetAdenosine kinase(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50350195(CHEMBL1814763)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human ADK using [3H]-adenosine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1CQXPubMed
TargetAdenosine kinase(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50350199(CHEMBL1814767)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human ADK using [3H]-adenosine by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1CQXPubMed
TargetThymidine phosphorylase(Escherichia coli)
Academy of Sciences of the Czech Republic

LigandPNGBDBM20033(6-(azetidin-1-yl)-5-bromo-1,3-diazinane-2,4-dione ...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:The enzyme reaction was started by the addition of enzyme to the reaction mixture containing substrate and test compounds. The reaction was stopped b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4VCHPubMed
TargetAdenosine kinase(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50028657(CHEMBL1814778)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human ADK expressed in Escherichia coli BL21(DE3) cells using [3H]adenosine by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29888MKPubMed
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