Compile Data Set for Download or QSAR
Found 383 with Last Name = 'lemasson' and Initial = 'ia'
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357011(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356996(5-Amino-N-(4-chloro-2-fluoro-phenyl)-1-(o-tolyl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357006(5-Amino-3-ethyl-1-(3-fluoro-2-methylphenyl)-N-[5-t...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357010(5-Amino-1-(2-hydroxyphenyl)-N-(5-(trifluoromethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357002(5-Amino-3-ethyl-1-(2-methoxyphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357007(5-Amino-1-(2-fluorophenyl)-3-methyl-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356998(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357004(5-Amino-N-(5-chloro-2-pyridyl)-1-(3-fluoro-2-methy...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356997(5-Amino-N-(2-fluoro-4-(trifluoromethyl)phenyl)-1-(...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357008(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357003(5-Amino-1-(2-(2-methoxyethoxy)phenyl)-3-methyl-N-(...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356995(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357001(5-Amino-N-(5-chloropyridin-2-yl)-1-(3-fluoro-2-met...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356999((5-Amino-1-(3-fluoro-2-methylphenyl)-1H-pyrazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357000((5-Amino-1-(2-methoxyphenyl)-1H-pyrazol-4-yl)(5-ch...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357009(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(2-methoxypy...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357005(5-Amino-1-(2-ethylphenyl)-N-(5-(2,2,2-trifluoroeth...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357012(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357006(5-Amino-3-ethyl-1-(3-fluoro-2-methylphenyl)-N-[5-t...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357008(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356995(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357000((5-Amino-1-(2-methoxyphenyl)-1H-pyrazol-4-yl)(5-ch...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357004(5-Amino-N-(5-chloro-2-pyridyl)-1-(3-fluoro-2-methy...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357002(5-Amino-3-ethyl-1-(2-methoxyphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357001(5-Amino-N-(5-chloropyridin-2-yl)-1-(3-fluoro-2-met...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357007(5-Amino-1-(2-fluorophenyl)-3-methyl-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356999((5-Amino-1-(3-fluoro-2-methylphenyl)-1H-pyrazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356998(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357009(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(2-methoxypy...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356997(5-Amino-N-(2-fluoro-4-(trifluoromethyl)phenyl)-1-(...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357010(5-Amino-1-(2-hydroxyphenyl)-N-(5-(trifluoromethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM356996(5-Amino-N-(4-chloro-2-fluoro-phenyl)-1-(o-tolyl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357005(5-Amino-1-(2-ethylphenyl)-N-(5-(2,2,2-trifluoroeth...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357003(5-Amino-1-(2-(2-methoxyethoxy)phenyl)-3-methyl-N-(...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Almirall, S.A.

US Patent
LigandPNGBDBM357012(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FQ9ZWJUS Patent
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Laboratoire de Chimie et de Biochimie Pharmacologiques et Toxicologiques , CNRS UMR 8601, Université Paris Descartes, Sorbonne Paris Cité , 45 rue des Saints-Pères , 75270 Paris Cedex 06 , France.

Curated by ChEMBL
LigandPNGBDBM50446782(CHEMBL3114672)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+6nMAssay Description:Antagonist activity at rat GluN1a/GluN2A receptors expressed in Xenopus laevis oocytes assessed as inhibition of L-glutamate/glucine induced current ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0BR0PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(RAT)
Laboratoire de Chimie et de Biochimie Pharmacologiques et Toxicologiques , CNRS UMR 8601, Université Paris Descartes, Sorbonne Paris Cité , 45 rue des Saints-Pères , 75270 Paris Cedex 06 , France.

Curated by ChEMBL
LigandPNGBDBM50446782(CHEMBL3114672)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+6nMAssay Description:Antagonist activity at rat GluN1a/mouse GluN2B receptors expressed in Xenopus laevis oocytes assessed as inhibition of L-glutamate/glucine induced cu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0BR0PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314793((S)-3-amino-3-carboxypropyl-2'-carboxyethyl phosph...)copy SMILEScopy InChI
Affinity DataEC50:  5.20E+4nMAssay Description:Agonist activity at rat mGlu2 receptor expressed in HEK293 cells assessed as increase in intracellular calcium level after 1 hr by fluorescence micro...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314794((3S)-2-[((3-Amino-3-carboxy)propyl)(hydroxy)phosph...)copy SMILEScopy InChI
Affinity DataEC50:  5.70E+4nMAssay Description:Agonist activity at rat mGlu2 receptor expressed in HEK293 cells assessed as increase in intracellular calcium level after 1 hr by fluorescence micro...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314796((3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosph...)copy SMILEScopy InChI
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at rat mGlu2 receptor expressed in HEK293 cells assessed as increase in intracellular calcium level after 1 hr by fluorescence micro...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314797((3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosph...)copy SMILEScopy InChI
Affinity DataEC50:  4.90E+4nMAssay Description:Agonist activity at rat mGlu2 receptor expressed in HEK293 cells assessed as increase in intracellular calcium level after 1 hr by fluorescence micro...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50034503((1R,2R)-3-((S)-Amino-carboxy-methyl)-cyclopropane-...)copy SMILEScopy InChI
Affinity DataEC50:  45nMAssay Description:Agonist activity at rat mGlu2 receptor expressed in HEK293 cells assessed as increase in intracellular calcium level after 1 hr by fluorescence micro...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314797((3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosph...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat mGlu7 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)copy SMILEScopy InChI
Affinity DataEC50:  3.06E+5nMAssay Description:Agonist activity at rat mGlu7 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50060137((1R,2S)-4-aminocyclopentane-1,2,4-tricarboxylic ac...)copy SMILEScopy InChI
Affinity DataEC50:  2.80E+5nMAssay Description:Agonist activity at rat mGlu7 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Agonist activity at rat mGlu8 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314793((S)-3-amino-3-carboxypropyl-2'-carboxyethyl phosph...)copy SMILEScopy InChI
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at rat mGlu8 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314794((3S)-2-[((3-Amino-3-carboxy)propyl)(hydroxy)phosph...)copy SMILEScopy InChI
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at rat mGlu8 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314795((3S)-4-[((3-Amino-3-carboxy)propyl)(hydroxy)phosph...)copy SMILEScopy InChI
Affinity DataEC50:  1.80E+4nMAssay Description:Agonist activity at rat mGlu8 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Universite Paris Descartes

Curated by ChEMBL
LigandPNGBDBM50314796((3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosph...)copy SMILEScopy InChI
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at rat mGlu8 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3F7QPubMed
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