Compile Data Set for Download or QSAR
Found 195 with Last Name = 'stroke' and Initial = 'il'
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454459(CHEMBL4215036)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454459(CHEMBL4215036)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507130(CHEMBL4452983)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507108(CHEMBL4529863)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454498(CHEMBL4215657)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454497(CHEMBL4214079)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454500(CHEMBL4212258)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507128(CHEMBL4451752)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507134(CHEMBL4444965)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507115(CHEMBL4520413)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507107(CHEMBL4473557)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507135(CHEMBL4470638)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507120(CHEMBL4473443)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507105(CHEMBL4557223)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507127(CHEMBL4476228)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507133(CHEMBL4461315)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507136(CHEMBL4454294)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454497(CHEMBL4214079)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507126(CHEMBL4483028)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507114(CHEMBL4553525)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507113(CHEMBL4436890)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454486(CHEMBL4203819)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507116(CHEMBL4452876)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507119(CHEMBL4441033)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507106(CHEMBL4472977)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507129(CHEMBL4456814)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507112(CHEMBL4547929)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454504(CHEMBL4210388)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Pharmacopeia, Inc.

Curated by ChEMBL
LigandPNGBDBM50413094(CHEMBL486116)copy SMILEScopy InChI
Affinity DataIC50: 18.6nMAssay Description:Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082N5PubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Pharmacopeia, Inc.

Curated by ChEMBL
LigandPNGBDBM50413093(CHEMBL528990)copy SMILEScopy InChI
Affinity DataIC50: 19.5nMAssay Description:Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082N5PubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery, Inc.

Curated by ChEMBL
LigandPNGBDBM50175173(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of CXCL10(IP-10)-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94GDPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507118(CHEMBL4456808)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507117(CHEMBL4591470)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507105(CHEMBL4557223)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Pharmacopeia, Inc.

Curated by ChEMBL
LigandPNGBDBM50413092(CHEMBL519258)copy SMILEScopy InChI
Affinity DataIC50: 25.1nMAssay Description:Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082N5PubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507135(CHEMBL4470638)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507109(CHEMBL4530206)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507121(CHEMBL4589634)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454503(CHEMBL4211420)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454498(CHEMBL4215657)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507110(CHEMBL4545776)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454502(CHEMBL4209041)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR50RGPubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery, Inc.

Curated by ChEMBL
LigandPNGBDBM50175193(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94GDPubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Pharmacopeia, Inc.

Curated by ChEMBL
LigandPNGBDBM50413100(CHEMBL485915)copy SMILEScopy InChI
Affinity DataIC50: 51.3nMAssay Description:Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082N5PubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507114(CHEMBL4553525)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507115(CHEMBL4520413)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP85FQPubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery, Inc.

Curated by ChEMBL
LigandPNGBDBM50175183(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94GDPubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery, Inc.

Curated by ChEMBL
LigandPNGBDBM50175168(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94GDPubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery, Inc.

Curated by ChEMBL
LigandPNGBDBM50175176(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-fluor...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94GDPubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery, Inc.

Curated by ChEMBL
LigandPNGBDBM50175173(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94GDPubMed
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