Compile Data Set for Download or QSAR
Found 16 with Last Name = 'windsor' and Initial = 'iw'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50505279(CHEMBL4436207)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:In vitro inhibitory effect of histamine H3 antagonist on the electrically evoked contractile response of isolated guinea pig jejunum segments.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM8125((3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl N-[(2S...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:In vitro inhibitory effect of histamine H3 antagonist on the electrically evoked contractile response of isolated guinea pig jejunum segments.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50406170(CHEMBL5266997)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:In vitro inhibitory effect of histamine H3 antagonist on the electrically evoked contractile response of isolated guinea pig jejunum segments.More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241605(CHEMBL4082603)copy SMILEScopy InChI
Affinity DataKd:  990nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50197883(CHEBI:78538 | FX-1006 | Tafamidis | US10377729, Co...)copy SMILEScopy InChI
Affinity DataKd:  278nMAssay Description:Binding affinity to wild type TTR (unknown origin) assessed as equilibrium dissociation constant of second site by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241609(CHEMBL4102478)copy SMILEScopy InChI
Affinity DataKd:  820nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9D7ZPubMed
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241612(CHEMBL4078202)copy SMILEScopy InChI
Affinity DataKd:  470nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50197883(CHEBI:78538 | FX-1006 | Tafamidis | US10377729, Co...)copy SMILEScopy InChI
Affinity DataKd:  370nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241613(CHEMBL4090439)copy SMILEScopy InChI
Affinity DataKd:  450nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241614(CHEMBL4069407)copy SMILEScopy InChI
Affinity DataKd:  470nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241615(CHEMBL4065175)copy SMILEScopy InChI
Affinity DataKd:  790nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9D7ZPubMed
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)copy SMILEScopy InChI
Affinity DataKd:  470nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241604(CHEMBL4060726)copy SMILEScopy InChI
Affinity DataKd:  1.80E+3nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241603(CHEMBL4072121)copy SMILEScopy InChI
Affinity DataKd:  440nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241598(CHEMBL4063503)copy SMILEScopy InChI
Affinity DataKd:  470nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50241602(CHEMBL4099088)copy SMILEScopy InChI
Affinity DataKd:  730nMAssay Description:Competitive binding affinity to human wild type TTR expressed in Escherichia coli BL-21 assessed as equilibrium dissociation constant of second site ...More data for this Ligand-Target Pair