Compile Data Set for Download or QSAR
Found 198 with Last Name = 'camacho' and Initial = 'j'
TargetEstrogen receptor(Homo sapiens (Human))
Instituto Politécnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)copy SMILEScopy InChI
Affinity DataKi:  0.160nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128311(US8796284, 93)copy SMILEScopy InChI
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128297(US8796284, 4)copy SMILEScopy InChI
Affinity DataKi:  6nM ΔG°:  -46.9kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128310(US8796284, 48)copy SMILEScopy InChI
Affinity DataKi:  7nM ΔG°:  -46.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128307(US8796284, 38)copy SMILEScopy InChI
Affinity DataKi:  7nM ΔG°:  -46.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128306(US8796284, 36)copy SMILEScopy InChI
Affinity DataKi:  8nM ΔG°:  -46.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128305(US8796284, 29)copy SMILEScopy InChI
Affinity DataKi:  10nM ΔG°:  -45.7kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128296(US8796284, 3)copy SMILEScopy InChI
Affinity DataKi:  11nM ΔG°:  -45.4kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128295(US8796284, 1)copy SMILEScopy InChI
Affinity DataKi:  12nM ΔG°:  -45.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375232(3-chloro-5-(3-fluoropyridin-4-yl)-6-(pyridin-4-yl)...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128311(US8796284, 93)copy SMILEScopy InChI
Affinity DataKi:  12nM ΔG°:  -47.0kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375233(3-bromo-5-(3-fluoropyridin-4-yl)-6-(pyridin-4-yl)p...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetEstrogen receptor(Homo sapiens (Human))
Instituto Politécnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323914(CHEMBL1213786 | Tamoxifen butyl bromide)copy SMILEScopy InChI
Affinity DataKi:  13.0nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QT9PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Instituto Politécnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323912(CHEMBL1213784 | Tamoxifen ethyl bromide)copy SMILEScopy InChI
Affinity DataKi:  13.7nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QT9PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128303(US8796284, 20)copy SMILEScopy InChI
Affinity DataKi:  14nM ΔG°:  -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128298(US8796284, 5)copy SMILEScopy InChI
Affinity DataKi:  14nM ΔG°:  -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128308(US8796284, 44)copy SMILEScopy InChI
Affinity DataKi:  14nM ΔG°:  -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128304(US8796284, 24)copy SMILEScopy InChI
Affinity DataKi:  16nM ΔG°:  -44.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128309(US8796284, 46)copy SMILEScopy InChI
Affinity DataKi:  17nM ΔG°:  -44.3kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128299(US8796284, 8)copy SMILEScopy InChI
Affinity DataKi:  18nM ΔG°:  -44.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128301(US8796284, 10)copy SMILEScopy InChI
Affinity DataKi:  21nM ΔG°:  -43.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375229(3-chloro-5-(3-fluoropyridin-4-yl)-6-(pyridin-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  23.9nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375234(3-chloro-5-(3-fluoropyridin-4-yl)-6-(6-methoxypyri...)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128295(US8796284, 1)copy SMILEScopy InChI
Affinity DataKi:  25nM ΔG°:  -45.1kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetEstrogen receptor(Homo sapiens (Human))
Instituto Politécnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323913(CHEMBL1213785 | Tamoxifen isopropyl bromide)copy SMILEScopy InChI
Affinity DataKi:  25.4nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QT9PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458396(US10744125, Example 5)copy SMILEScopy InChI
Affinity DataKi:  26.3nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458398(US10744125, Example 14)copy SMILEScopy InChI
Affinity DataKi:  29.2nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetEstrogen receptor(Homo sapiens (Human))
Instituto Politécnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)copy SMILEScopy InChI
Affinity DataKi:  31.2nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QT9PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128300(US8796284, 9)copy SMILEScopy InChI
Affinity DataKi:  33nM ΔG°:  -42.7kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375227(3-chloro-6-(pyridin-3-yl)-5-(pyridin-4-yl)pyridin-...)copy SMILEScopy InChI
Affinity DataKi:  34.5nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128302(US8796284, 13)copy SMILEScopy InChI
Affinity DataKi:  35nM ΔG°:  -42.6kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375230(3-bromo-5-(3-fluoropyridin-4-yl)-6-(pyridin-3-yl)p...)copy SMILEScopy InChI
Affinity DataKi:  37nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375228(3-bromo-6-(pyridin-3-yl)-5-(pyridin-4-yl)pyridin-2...)copy SMILEScopy InChI
Affinity DataKi:  46.1nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetEstrogen receptor(Homo sapiens (Human))
Instituto Politécnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323911(CHEMBL1213783 | Tamoxifen methyl iodide)copy SMILEScopy InChI
Affinity DataKi:  46.3nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QT9PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458394(US10744125, Example 4)copy SMILEScopy InChI
Affinity DataKi:  47.6nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128302(US8796284, 13)copy SMILEScopy InChI
Affinity DataKi:  50nM ΔG°:  -43.3kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458397(US10744125, Example 6)copy SMILEScopy InChI
Affinity DataKi:  50.3nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM128299(US8796284, 8)copy SMILEScopy InChI
Affinity DataKi:  60nM ΔG°:  -42.9kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WM1C2QUS Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458392(US10744125, Example 3)copy SMILEScopy InChI
Affinity DataKi:  65.5nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458389(US10744125, Example 1)copy SMILEScopy InChI
Affinity DataKi:  103nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375226(5-(3-fluoropyridin-4-yl)-6-(pyridin-4-yl)pyridin-2...)copy SMILEScopy InChI
Affinity DataKi:  149nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM375231(3-chloro-6-(5-fluoropyridin-3-yl)-5-(3-fluoropyrid...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM375228(3-bromo-6-(pyridin-3-yl)-5-(pyridin-4-yl)pyridin-2...)copy SMILEScopy InChI
Affinity DataKi:  300nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458389(US10744125, Example 1)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM458389(US10744125, Example 1)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM375227(3-chloro-6-(pyridin-3-yl)-5-(pyridin-4-yl)pyridin-...)copy SMILEScopy InChI
Affinity DataKi:  500nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP48FVUS Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458398(US10744125, Example 14)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458398(US10744125, Example 14)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:A2A Adenosine Receptor: Competitive assays were carried out by incubation of membranes from human A2A receptors transfected to HeLa cells, [3H]-ZM241...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vanderbilt University School of Medicine

LigandPNGBDBM458396(US10744125, Example 5)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Palobiofarma, S.L.

US Patent
LigandPNGBDBM458396(US10744125, Example 5)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F192SJUS Patent
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