Affinity DataKi: 0.160nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -51.4kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 6nM ΔG°: -46.9kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 7nM ΔG°: -46.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 7nM ΔG°: -46.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 8nM ΔG°: -46.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 10nM ΔG°: -45.7kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 11nM ΔG°: -45.4kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 12nM ΔG°: -45.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 12nM ΔG°: -47.0kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 13.0nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 13.7nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 14nM ΔG°: -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 14nM ΔG°: -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 14nM ΔG°: -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 16nM ΔG°: -44.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 17nM ΔG°: -44.3kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 18nM ΔG°: -44.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 21nM ΔG°: -43.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 23.9nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 25nM ΔG°: -45.1kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
Affinity DataKi: 25.4nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 26.3nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Affinity DataKi: 29.2nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Affinity DataKi: 31.2nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 33nM ΔG°: -42.7kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 34.5nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 35nM ΔG°: -42.6kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 46.1nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 46.3nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 47.6nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Affinity DataKi: 50nM ΔG°: -43.3kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
Affinity DataKi: 50.3nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Affinity DataKi: 60nM ΔG°: -42.9kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
Affinity DataKi: 65.5nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:A3 Adenosine Receptor:Competitive assays were carried out by incubation of membranes from human A3 receptors transfected to CHO cells, [3H]-NECA, buf...More data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:A2A Adenosine Receptor: Competitive assays were carried out by incubation of membranes from human A2A receptors transfected to HeLa cells, [3H]-ZM241...More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:A2B Adenosine Receptor: The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCP...More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:Adenosine A1 Receptor: Competition assays were carried out by incubation of human recombinant membranes of adenosine receptors from hA1 receptors tra...More data for this Ligand-Target Pair