Compile Data Set for Download or QSAR
Found 143 with Last Name = 'cidado' and Initial = 'j'
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454567(US10717746, Example 48)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454570(US10717746, Example 51)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454542(US10717746, Example 25 | US10717746, Example 84)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454563(US10717746, Example 44)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454570(US10717746, Example 51)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454539(US10717746, Example 22)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50549515(CHEMBL4759074)copy SMILES
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454597(US10717746, Example 82)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM454542(US10717746, Example 25 | US10717746, Example 84)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK3 (unknown origin) in presence of 5 mM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454566(US10717746, Example 47)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454584(US10717746, Example 66)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of CDK3 (unknown origin) in presence of 5 mM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454544(US10717746, Example 27)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454542(US10717746, Example 25 | US10717746, Example 84)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454559(US10717746, Example 40 | US10717746, Example 41)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454559(US10717746, Example 40 | US10717746, Example 41)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454533(US10717746, Example 16)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM164883(US9067888, 33)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454539(US10717746, Example 22)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454559(US10717746, Example 40 | US10717746, Example 41)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454519(US10717746, Example 2)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454566(US10717746, Example 47)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454567(US10717746, Example 48)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454544(US10717746, Example 27)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454563(US10717746, Example 44)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50549515(CHEMBL4759074)copy SMILES
Affinity DataIC50: 49nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454582(US10717746, Example 63)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
LigandPNGBDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of recombinant full length human CDK2/CyclinE expressed in insect cells using FL-Ahx-QSPKKG-CONH2 as substrate preincubated for 10 mins fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454593(US10717746, Example 78)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50549519(CHEMBL4759053)copy SMILES
Affinity DataIC50: 61nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454558(US10717746, Example 39)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
LigandPNGBDBM454542(US10717746, Example 25 | US10717746, Example 84)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant full length human CDK2/CyclinE expressed in insect cells using FL-Ahx-QSPKKG-CONH2 as substrate preincubated for 10 mins fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454559(US10717746, Example 40 | US10717746, Example 41)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM454519(US10717746, Example 2)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of CDK3 (unknown origin) in presence of 5 mM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454594(US10717746, Example 78a)copy SMILES
Affinity DataIC50: 85nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454584(US10717746, Example 66)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
LigandPNGBDBM454542(US10717746, Example 25 | US10717746, Example 84)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Inhibition of recombinant full length human His-tagged CDK1/CyclinB expressed in baculovirus infected insect cells using 5FAM-RRRFRPASPLRGPPKCOOH as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454582(US10717746, Example 63)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454525(US10717746, Example 8)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454519(US10717746, Example 2)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
LigandPNGBDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)copy SMILEScopy InChI
Affinity DataIC50: 117nMAssay Description:Inhibition of recombinant full length human His-tagged CDK1/CyclinB expressed in baculovirus infected insect cells using 5FAM-RRRFRPASPLRGPPKCOOH as ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM164883(US9067888, 33)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454598(US10717746, Example 82a)copy SMILES
Affinity DataIC50: 139nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50549519(CHEMBL4759053)copy SMILES
Affinity DataIC50: 140nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454558(US10717746, Example 39)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454533(US10717746, Example 16)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454597(US10717746, Example 82)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser2 residues measured after 6 hrs by immunof...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM454527(US10717746, Example 10)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant full length human N-terminal GST-fused CDK9 (1 to 372 residues)/His-tagged CyclinT1 (1 to 726 residues) expressed in baculo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
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