Compile Data Set for Download or QSAR
Found 127 with Last Name = 'dell-john' and Initial = 'j'
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122646(CHEMBL3623125)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122650(CHEMBL3623127)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122647(CHEMBL3623126)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122640(CHEMBL3623119)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323038(4-[(1S,2S,6R,7R)-9-(6-Chloro-pyrimidin-4-yl)-1,7-d...)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323017(4-((1S,2S,6R,7R)-9-Methoxy-1,7-dimethyl-3,5-dioxo-...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323023((1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phenyl)...)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323039(4-((1S,2S,6R,7R)-1,7-Dimethyl-3,5-dioxo-9-pyrimidi...)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323024((1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phenyl)...)copy SMILEScopy InChI
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122643(CHEMBL3623122)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122635(CHEMBL3623114)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323035(3-[(1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phen...)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323037(4-[(1S,2S,6R,7R)-9-(3-Methanesulfonyl-phenyl)-1,7-...)copy SMILEScopy InChI
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122645(CHEMBL3623124)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323025((1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phenyl)...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122644(CHEMBL3623123)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323032(4-[(1R,2R,6S,7S)-3,5-dioxo-9-(phenylsulfonyl)-11-o...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323018(4-((1S,2S,6R,7R)-1,7-Dimethyl-3,5-dioxo-9-propyl-1...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323015(4-((1S,2S,6R,7R)-9-Isopropyl-1,7-dimethyl-3,5,8,10...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323031(4-((1S,2S,6R,7R)-9-Ethanesulfonyl-1,7-dimethyl-3,5...)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323012(2-Trifluoromethyl-4-((1S,2S,6R,7R)-1,7,9-trimethyl...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323011(4-((1S,2S,6R,7R)-1,7-Dimethyl-3,5-dioxo-11-oxa-4,9...)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323036(3-[(1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phen...)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323022(4-((1S,2S,6R,7R)-9-Benzoyl-1,7-dimethyl-3,5-dioxo-...)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122637(CHEMBL3623116)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323029((1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phenyl)...)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122639(CHEMBL3623118)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122642(CHEMBL3623121)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323033(4-[(1S,2S,6R,7R)-9-(4-Fluoro-benzenesulfonyl)-1,7-...)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323021(4-((1S,2S,6R,7R)-9-Cyclopropanecarbonyl-1,7-dimeth...)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323016(4-((1S,2S,6R,7R)-9-Hydroxy-1,7-dimethyl-3,5-dioxo-...)copy SMILEScopy InChI
Affinity DataKi:  37nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323020(4-((1S,2S,6R,7R)-9-Isobutyryl-1,7-dimethyl-3,5-dio...)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323028((1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phenyl)...)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323013(4-((1S,2S,6R,7R)-9-Cyclopropylmethyl-1,7-dimethyl-...)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122638(CHEMBL3623117)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122641(CHEMBL3623120)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323030(4-((1S,2S,6R,7R)-9-Methanesulfonyl-1,7-dimethyl-3,...)copy SMILEScopy InChI
Affinity DataKi:  56nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)copy SMILEScopy InChI
Affinity DataKi:  64nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)copy SMILEScopy InChI
Affinity DataKi:  64nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323019(4-[(1R,2R,6S,7S)-3,5-dioxo-9-propionyl-11-oxa-4,9-...)copy SMILEScopy InChI
Affinity DataKi:  84nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323034(4-[(1S,2S,6R,7R)-1,7-Dimethyl-3,5-dioxo-9-(pyridin...)copy SMILEScopy InChI
Affinity DataKi:  93nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323027((1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phenyl)...)copy SMILEScopy InChI
Affinity DataKi:  98nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323026((1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phenyl)...)copy SMILEScopy InChI
Affinity DataKi:  176nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122636(CHEMBL3623115)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323014(4-((1S,2S,6R,7R)-9-Isopropyl-1,7-dimethyl-3,5,8,10...)copy SMILEScopy InChI
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [3H]DHT from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122645(CHEMBL3623124)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122643(CHEMBL3623122)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50122647(CHEMBL3623126)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase repor...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3P96PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323037(4-[(1S,2S,6R,7R)-9-(3-Methanesulfonyl-phenyl)-1,7-...)copy SMILEScopy InChI
Affinity DataIC50: 7.40nMAssay Description:Antagonist activity at human wild type AR expressed in human MDA-MB-435 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol Myers-Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50323035(3-[(1S,2S,6R,7R)-4-(4-Cyano-3-trifluoromethyl-phen...)copy SMILEScopy InChI
Affinity DataIC50: 7.40nMAssay Description:Antagonist activity at human wild type AR expressed in human MDA-MB-435 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6DVHPubMed
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