Compile Data Set for Download or QSAR
Found 141 with Last Name = 'eickhoff' and Initial = 'j'
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Merck Patent GmbH

US Patent
LigandPNGBDBM251929(US9481668, A6)copy SMILEScopy InChI
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The kinase assay was carried out as 384-well FlashPlate assay. As test plates 384-well streptavidine coated FlashPlate microtitre plates from Perkin ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26H4GBFUS Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509371(CHEMBL4521241)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
Target14-3-3 protein sigma(Homo sapiens (Human))
Eindhoven University of Technology

Curated by ChEMBL
LigandPNGBDBM50462085(CHEMBL4240436)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TMR-GG-RLSHpSSLPG-NH2 binding to recombinant human GST-tagged 14-3-3-sigma preincubated for 30 mins followed by TMR-GG-RLSHpSSLPG-NH2 a...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB7781PubMed
Target14-3-3 protein sigma(Homo sapiens (Human))
Eindhoven University of Technology

Curated by ChEMBL
LigandPNGBDBM50462084(CHEMBL4247540)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TMR-GG-RLSHpSSLPG-NH2 binding to recombinant human GST-tagged 14-3-3-sigma preincubated for 30 mins followed by TMR-GG-RLSHpSSLPG-NH2 a...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB7781PubMed
Target14-3-3 protein sigma(Homo sapiens (Human))
Eindhoven University of Technology

Curated by ChEMBL
LigandPNGBDBM50462083(CHEMBL4237531)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TMR-GG-RLSHpSSLPG-NH2 binding to recombinant human GST-tagged 14-3-3-sigma preincubated for 30 mins followed by TMR-GG-RLSHpSSLPG-NH2 a...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB7781PubMed
Target14-3-3 protein sigma(Homo sapiens (Human))
Eindhoven University of Technology

Curated by ChEMBL
LigandPNGBDBM50462080(CHEMBL4250552)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TMR-GG-RLSHpSSLPG-NH2 binding to recombinant human GST-tagged 14-3-3-sigma preincubated for 30 mins followed by TMR-GG-RLSHpSSLPG-NH2 a...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB7781PubMed
Target14-3-3 protein sigma(Homo sapiens (Human))
Eindhoven University of Technology

Curated by ChEMBL
LigandPNGBDBM50462078(CHEMBL4243744)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TMR-GG-RLSHpSSLPG-NH2 binding to recombinant human GST-tagged 14-3-3-sigma preincubated for 30 mins followed by TMR-GG-RLSHpSSLPG-NH2 a...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB7781PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153641(US8999982, Ref4)copy SMILEScopy InChI
Affinity DataIC50: 7.04E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)copy SMILEScopy InChI
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153643(US8999982, Ref6)copy SMILEScopy InChI
Affinity DataIC50: 8.29E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153652(US8999982, 3-fluoro-4-((6-methoxy-7-(3- morpholino...)copy SMILEScopy InChI
Affinity DataIC50: 8.50E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
Target14-3-3 protein zeta/delta(Homo sapiens)
Eindhoven University of Technology

Curated by ChEMBL
LigandPNGBDBM50102295(4-(4-Formyl-5-hydroxy-6-methyl-3-phosphonooxymethy...)copy SMILEScopy InChI
Affinity DataIC50: 9.30E+3nMAssay Description:Binding affinity to GST-tagged 14-3-3-zeta (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as inhibition of interaction with PRAS40...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153644(US8999982, Ref7)copy SMILEScopy InChI
Affinity DataIC50: 9.30E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK2 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM50317324(CHEMBL1087984 | N-(4-(6,7-dimethoxyquinolin-4-ylox...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153639(US8999982, Ref2)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153640(US8999982, Ref3)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153642(US8999982, Ref5)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153645(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153646(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)ani...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153647(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153648(US8999982, 3-chloro-4-((6,7- dimethoxyquinolin-4- ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153649(US8999982, 5-((6,7-dimethoxyquinolin-4- yl)oxy)pyr...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153650(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153651(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Lead Discovery Center GmbH; Max-Planck-Gesellschaft zur Förderung der Wissenschaften E.V.

US Patent
LigandPNGBDBM153653(US8999982, tert-butyl 4-(((4-(4-amino-2- fluorophe...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SQ8Z4DUS Patent
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