Compile Data Set for Download or QSAR
Found 302 with Last Name = 'falcone' and Initial = 'j'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)copy SMILEScopy InChI
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMedDrugBank
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1BZZPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)copy SMILEScopy InChI
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1BZZPubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1BZZPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1BZZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
TargetD(1A) dopamine receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)copy SMILEScopy InChI
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetHistamine H1 receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetAlpha-2C adrenergic receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetAlpha-2C adrenergic receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetD(1A) dopamine receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetHistamine H1 receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMedDrugBank
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetHistamine H1 receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
TargetHistamine H1 receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50095890(2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperaz...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetAlpha-2C adrenergic receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)copy SMILEScopy InChI
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4N5NPubMed
TargetHistamine H1 receptor(RAT)
Lilly Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50095890(2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperaz...)copy SMILEScopy InChI
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K1MPubMed
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