Compile Data Set for Download or QSAR
Found 840 with Last Name = 'fells' and Initial = 'j'
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50271765(3-(4-{3-[4-(3-Carboxy-acryloylamino)-phenoxy]-phen...)copy SMILEScopy InChI
Affinity DataKi:  7.20nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270817CPubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50271763(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)copy SMILEScopy InChI
Affinity DataKi:  20.8nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270817CPubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50271764(3-[4'-(3-Carboxy-acryloylamino)-biphenyl-4-ylcarba...)copy SMILEScopy InChI
Affinity DataKi:  21.1nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270817CPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50304580(2-(3-(4-nitrophenoxy)phenyl)-1,3-dioxoisoindoline-...)copy SMILEScopy InChI
Affinity DataKi:  48nMAssay Description:Binding affinity to LPA1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB244MPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50271763(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270817CPubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50304580(2-(3-(4-nitrophenoxy)phenyl)-1,3-dioxoisoindoline-...)copy SMILEScopy InChI
Affinity DataKi:  230nMAssay Description:Binding affinity to LPA3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB244MPubMed
TargetLysophosphatidic acid receptor 5(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50304580(2-(3-(4-nitrophenoxy)phenyl)-1,3-dioxoisoindoline-...)copy SMILEScopy InChI
Affinity DataKi:  292nMAssay Description:Binding affinity to LPA5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB244MPubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50271765(3-(4-{3-[4-(3-Carboxy-acryloylamino)-phenoxy]-phen...)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270817CPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50304581(2-(1,3-dioxo-5-(p-tolyloxy)isoindolin-2-yl)acetic ...)copy SMILEScopy InChI
Affinity DataKi:  311nMAssay Description:Binding affinity to LPA1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB244MPubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50241460(4-(3-benzamidophenylamino)-4-oxobut-2-enoic acid |...)copy SMILEScopy InChI
Affinity DataKi:  317nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270817CPubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50304581(2-(1,3-dioxo-5-(p-tolyloxy)isoindolin-2-yl)acetic ...)copy SMILEScopy InChI
Affinity DataKi:  1.08E+3nMAssay Description:Binding affinity to LPA3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB244MPubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50271764(3-[4'-(3-Carboxy-acryloylamino)-biphenyl-4-ylcarba...)copy SMILEScopy InChI
Affinity DataKi:  7.02E+3nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270817CPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University of Memphis

Curated by ChEMBL
LigandPNGBDBM50271765(3-(4-{3-[4-(3-Carboxy-acryloylamino)-phenoxy]-phen...)copy SMILEScopy InChI
Affinity DataKi:  1.35E+4nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q270817CPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50568214(CHEMBL4860000)copy SMILES
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR51V7PubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50544215(CHEMBL4637689)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0S85PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50544211(CHEMBL4641682)copy SMILEScopy InChI
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC1 expressed in HEK293F cells using FLUOR DE LYS as substrate preincubated for 3 hrs follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0S85PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50543650(CHEMBL4649205)copy SMILEScopy InChI
Affinity DataIC50: 0.0850nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50544211(CHEMBL4641682)copy SMILEScopy InChI
Affinity DataIC50: 0.0870nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0S85PubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50543650(CHEMBL4649205)copy SMILEScopy InChI
Affinity DataIC50: 0.0930nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50568211(CHEMBL4876610)copy SMILES
Affinity DataIC50: 0.110nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR51V7PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50543649(CHEMBL4644038)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50568215(CHEMBL4878197)copy SMILES
Affinity DataIC50: 0.110nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR51V7PubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50568215(CHEMBL4878197)copy SMILES
Affinity DataIC50: 0.130nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR51V7PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50544215(CHEMBL4637689)copy SMILEScopy InChI
Affinity DataIC50: 0.160nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC1 expressed in HEK293F cells using FLUOR DE LYS as substrate preincubated for 3 hrs follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0S85PubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50544227(CHEMBL4634501)copy SMILEScopy InChI
Affinity DataIC50: 0.170nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC3/His6-tagged SMRT (1 to 899 residues) expressed in HEK293F cells using FLUOR DE LYS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0S85PubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50543649(CHEMBL4644038)copy SMILEScopy InChI
Affinity DataIC50: 0.180nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50543637(CHEMBL4642518)copy SMILEScopy InChI
Affinity DataIC50: 0.190nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50543637(CHEMBL4642518)copy SMILEScopy InChI
Affinity DataIC50: 0.190nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50544227(CHEMBL4634501)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of full length human recombinant FLAG-tagged HDAC1 expressed in HEK293F cells using FLUOR DE LYS as substrate preincubated for 3 hrs follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0S85PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50568214(CHEMBL4860000)copy SMILES
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR51V7PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50543647(CHEMBL4637357)copy SMILEScopy InChI
Affinity DataIC50: 0.220nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50543643(CHEMBL4642023)copy SMILEScopy InChI
Affinity DataIC50: 0.240nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50606543(CHEMBL5218926)copy SMILES
Affinity DataIC50: 0.280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50543640(CHEMBL4638264)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50543640(CHEMBL4638264)copy SMILEScopy InChI
Affinity DataIC50: 0.290nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ3BQCPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50606550(CHEMBL5220616)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50606548(CHEMBL5218918)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50606555(CHEMBL5220926)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50606556(CHEMBL5218854)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50606557(CHEMBL5219294)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50568207(CHEMBL4856631)copy SMILES
Affinity DataIC50: 0.300nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR51V7PubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50568207(CHEMBL4856631)copy SMILES
Affinity DataIC50: 0.300nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR51V7PubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50568207(CHEMBL4856631)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50606548(CHEMBL5218918)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50606555(CHEMBL5220926)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50606556(CHEMBL5218854)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50606557(CHEMBL5219294)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50606558(CHEMBL5219825)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50606559(CHEMBL5219875)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50606560(CHEMBL5220360)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58RGNPubMed
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