Compile Data Set for Download or QSAR
Found 100 with Last Name = 'gising' and Initial = 'j'
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetGenome polyprotein(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50326056((1S,3aR,6aS)-2-((S)-2-((S)-2-cyclohexyl-2-(pyrazin...)copy SMILEScopy InChI
Affinity DataKi:  3.90nMAssay Description:Inhibition of full-length HCV NS3 protease D168V mutantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V127T4PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600576(CHEMBL5177359)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600590(CHEMBL5207511)copy SMILES
Affinity DataKi:  4.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600586(CHEMBL5170220)copy SMILES
Affinity DataKi:  5.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600578(CHEMBL5176951)copy SMILES
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600591(CHEMBL5174301)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549529(CHEMBL4779819)copy SMILES
Affinity DataKi:  6.60nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549533(CHEMBL4779945)copy SMILES
Affinity DataKi:  7.60nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600575(CHEMBL5205769)copy SMILES
Affinity DataKi:  9.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549530(CHEMBL4788892)copy SMILES
Affinity DataKi:  9.30nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600572(CHEMBL5178838)copy SMILES
Affinity DataKi:  9.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600588(CHEMBL5201369)copy SMILES
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600573(CHEMBL5172324)copy SMILES
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600589(CHEMBL5202149)copy SMILES
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600580(CHEMBL5200734)copy SMILES
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600587(CHEMBL5176607)copy SMILES
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600574(CHEMBL5191241)copy SMILES
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600585(CHEMBL5196244)copy SMILES
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549528(CHEMBL4759641)copy SMILES
Affinity DataKi:  17nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600577(CHEMBL5181652)copy SMILES
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetGenome polyprotein(Hepatitis C Virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50142916((1S,4R,6S,14S,18R)-14-Cyclopentyloxycarbonylamino-...)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of full-length HCV NS3 protease R155K mutantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V127T4PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549526(CHEMBL4751226)copy SMILES
Affinity DataKi:  26nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600571(CHEMBL5179052)copy SMILES
Affinity DataKi:  29nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600579(CHEMBL5198739)copy SMILES
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600581(CHEMBL5188126)copy SMILES
Affinity DataKi:  35nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549527(CHEMBL4784233)copy SMILES
Affinity DataKi:  39nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549525(CHEMBL2086911)copy SMILES
Affinity DataKi:  48nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549532(CHEMBL4747530)copy SMILES
Affinity DataKi:  53nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetGenome polyprotein(Hepatitis C Virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50326056((1S,3aR,6aS)-2-((S)-2-((S)-2-cyclohexyl-2-(pyrazin...)copy SMILEScopy InChI
Affinity DataKi:  82nMAssay Description:Inhibition of full-length HCV NS3 protease R155K mutantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V127T4PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549531(CHEMBL4762752)copy SMILES
Affinity DataKi:  110nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetGenome polyprotein(Hepatitis C Virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50142916((1S,4R,6S,14S,18R)-14-Cyclopentyloxycarbonylamino-...)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of full-length HCV NS3 protease A156T mutantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V127T4PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600582(CHEMBL5208437)copy SMILES
Affinity DataKi:  130nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetGenome polyprotein(Hepatitis C Virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496213(CHEMBL3125634)copy SMILEScopy InChI
Affinity DataKi:  170nMAssay Description:Inhibition of full-length HCV NS3 protease A156T mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V127T4PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549534(CHEMBL4797684)copy SMILES
Affinity DataKi:  170nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600575(CHEMBL5205769)copy SMILES
Affinity DataKi:  180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetGenome polyprotein(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50142916((1S,4R,6S,14S,18R)-14-Cyclopentyloxycarbonylamino-...)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of full-length HCV NS3 protease D168V mutantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V127T4PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50030814(CHEMBL2086892)copy SMILEScopy InChI
Affinity DataKi:  270nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50549524(CHEMBL2086910)copy SMILES
Affinity DataKi:  280nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WRZPubMed
TargetGenome polyprotein(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496213(CHEMBL3125634)copy SMILEScopy InChI
Affinity DataKi:  320nMAssay Description:Inhibition of full-length HCV NS3 protease D168V mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V127T4PubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600576(CHEMBL5177359)copy SMILES
Affinity DataKi:  390nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600580(CHEMBL5200734)copy SMILES
Affinity DataKi:  400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600581(CHEMBL5188126)copy SMILES
Affinity DataKi:  410nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetGenome polyprotein(Hepatitis C Virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496213(CHEMBL3125634)copy SMILEScopy InChI
Affinity DataKi:  420nMAssay Description:Inhibition of full-length HCV NS3 protease R155K mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V127T4PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600583(CHEMBL5189691)copy SMILES
Affinity DataKi:  460nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600574(CHEMBL5191241)copy SMILES
Affinity DataKi:  460nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600584(CHEMBL5199606)copy SMILES
Affinity DataKi:  590nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600572(CHEMBL5178838)copy SMILES
Affinity DataKi:  620nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600579(CHEMBL5198739)copy SMILES
Affinity DataKi:  710nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50600573(CHEMBL5172324)copy SMILES
Affinity DataKi:  710nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2V1DPubMed
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