Compile Data Set for Download or QSAR
Found 248 with Last Name = 'grembecka' and Initial = 'j'
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMedMMDB
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetProthrombin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50117680(CHEMBL3613792)copy SMILEScopy InChI
Affinity DataKi:  57nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7J2HPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129685(2-Amino-4-methyl-pentanal | CHEMBL88476)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)copy SMILEScopy InChI
Affinity DataKi:  67nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129682(2-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoylme...)copy SMILEScopy InChI
Affinity DataKi:  74nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129679((1-Amino-3-methyl-butyl)-phosphonic acid | 1-amino...)copy SMILEScopy InChI
Affinity DataKi:  230nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)copy SMILEScopy InChI
Affinity DataKi:  276nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetProthrombin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50117692(CHEMBL3613791)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7J2HPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129677(3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl]-p...)copy SMILEScopy InChI
Affinity DataKi:  330nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129682(2-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoylme...)copy SMILEScopy InChI
Affinity DataKi:  1.01E+3nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)copy SMILEScopy InChI
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129677(3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl]-p...)copy SMILEScopy InChI
Affinity DataKi:  1.42E+3nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129680(CHEMBL423870 | {[hydroxy(1-hydroxy-3-methylbutyl)p...)copy SMILEScopy InChI
Affinity DataKi:  4.88E+3nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129679((1-Amino-3-methyl-butyl)-phosphonic acid | 1-amino...)copy SMILEScopy InChI
Affinity DataKi:  5.50E+4nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50129678(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyloxy...)copy SMILEScopy InChI
Affinity DataKi:  5.80E+4nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P903FPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455873(CHEMBL4216801)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455856(CHEMBL4218724)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455865(CHEMBL4211318)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455881(CHEMBL4204254)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455883(CHEMBL4207749)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455862(CHEMBL4207527)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455880(CHEMBL4209476)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455860(CHEMBL4203695)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetTubulin polymerization-promoting protein(Homo sapiens (Human))
University of Virginia

LigandPNGBDBM59225(Boronic acid, cis-6 | Boronic acid, trans-6)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:IC50 values for inhibition of cell growth using MCF-7 cell line were obtained by measuring the amount of total cell protein with the sulforhodamine B...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN43HCPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455864(CHEMBL4203028)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455868(CHEMBL4204241)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455861(CHEMBL4218853)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455879(CHEMBL4205576)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455874(CHEMBL4208216)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455869(CHEMBL4209696)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455859(CHEMBL3780895)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetTubulin polymerization-promoting protein(Homo sapiens (Human))
University of Virginia

LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:IC50 values for inhibition of cell growth using MCF-7 cell line were obtained by measuring the amount of total cell protein with the sulforhodamine B...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN43HCPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455876(CHEMBL4217916)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455872(CHEMBL4204591)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455863(CHEMBL4204941)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455884(CHEMBL4210554)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455867(CHEMBL4213678)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455858(CHEMBL4210798)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50117750(CHEMBL3586090)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of N-terminal thioredoxin His6-tagged full-length human menin expressed in Escherichia coli Rosetta (DE3) cells assessed as reduction in m...More data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455857(CHEMBL4218711)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50496327(CHEMBL3126198)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455882(CHEMBL4207176)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50455870(CHEMBL4210221)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03BRFPubMed
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50117744(CHEMBL3613789)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of N-terminal thioredoxin His6-tagged full-length human menin expressed in Escherichia coli Rosetta (DE3) cells assessed as reduction in m...More data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50496346(CHEMBL3126196)copy SMILEScopy InChI
Affinity DataIC50: 67nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
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