Compile Data Set for Download or QSAR
Found 162 with Last Name = 'habel' and Initial = 'j'
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303639(CHEMBL571626 | N-(4-(2-(4-(1H-1,2,3-Triazol-1-yl)p...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303638(4-(4-(4-(Methylsulfonamido)phenyl)pyrimidin-2-ylam...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM92524(Aminopyrazole inhibitor, 3576)copy SMILEScopy InChI
Affinity DataIC50: 7nMpH: 7.0 T: 2°CAssay Description:Homogeneous time-resolved fluorescence assay is an enzyme inhibition studies that were performed in 384-well polystyrene homogeneous time-resolved fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ867TPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303639(CHEMBL571626 | N-(4-(2-(4-(1H-1,2,3-Triazol-1-yl)p...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303638(4-(4-(4-(Methylsulfonamido)phenyl)pyrimidin-2-ylam...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM92523(Aminopyrazole inhibitor, 3528)copy SMILEScopy InChI
Affinity DataIC50: 23nMpH: 7.0 T: 2°CAssay Description:Homogeneous time-resolved fluorescence assay is an enzyme inhibition studies that were performed in 384-well polystyrene homogeneous time-resolved fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ867TPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM92522(Aminopyrazole inhibitor, 3451)copy SMILEScopy InChI
Affinity DataIC50: 25nMpH: 7.0 T: 2°CAssay Description:Homogeneous time-resolved fluorescence assay is an enzyme inhibition studies that were performed in 384-well polystyrene homogeneous time-resolved fl...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303644(3-Morpholino-5-(2-(4-(3-(pyridin-2-yl)-1H-1,2,4-tr...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32488(aryl piperidine, 9d)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303642(3-(2-(4-(2-Methyl-2H-tetrazol-5-yl)phenylamino)pyr...)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303641(3-(2-(4-(3-Methyl-1H-1,2,4-triazol-1-yl)phenylamin...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM92526(Aminopyrazole inhibitor, 4326)copy SMILEScopy InChI
Affinity DataIC50: 55nMpH: 7.0 T: 2°CAssay Description:Homogeneous time-resolved fluorescence assay is an enzyme inhibition studies that were performed in 384-well polystyrene homogeneous time-resolved fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ867TPubMed
TargetIsoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM32487(aryl piperidine, 9b)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303644(3-Morpholino-5-(2-(4-(3-(pyridin-2-yl)-1H-1,2,4-tr...)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303641(3-(2-(4-(3-Methyl-1H-1,2,4-triazol-1-yl)phenylamin...)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetIsoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM32488(aryl piperidine, 9d)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303643(4-(3-Morpholinophenyl)-N-(4-(3-(pyridin-3-yl)-1H-1...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32487(aryl piperidine, 9b)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303643(4-(3-Morpholinophenyl)-N-(4-(3-(pyridin-3-yl)-1H-1...)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303646(4-(3-Fluoro-5-morpholinophenyl)-N-(4-(3-morpholino...)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMedMMDB
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303645(4-(3-Fluoro-5-morpholinophenyl)-N-(4-(3-(4-methylp...)copy SMILEScopy InChI
Affinity DataIC50: 102nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32470(piperazine amide, 4q)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetIsoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM32494(aryl piperidine, 9j)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32494(aryl piperidine, 9j)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303640(CHEMBL585725 | N-(4-(3-Methyl-1H-1,2,4-triazol-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 113nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50169959(2-(benzo[d]thiazol-2(3H)-ylidene)-2-(2-(2-(pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of JNK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50224014(CHEMBL248983 | N-(4-(5-(5-chloropyridin-2-ylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of JNK3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36KXPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303637(CHEMBL572283 | N-(4-(1H-1,2,3-Triazol-1-yl)phenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:Inhibition of JNK1 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303645(4-(3-Fluoro-5-morpholinophenyl)-N-(4-(3-(4-methylp...)copy SMILEScopy InChI
Affinity DataIC50: 133nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50224001(CHEMBL248984 | N-(4-(5-(5-fluoropyridin-2-ylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of JNK3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36KXPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32460(piperazine amide, 4g)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303642(3-(2-(4-(2-Methyl-2H-tetrazol-5-yl)phenylamino)pyr...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50303646(4-(3-Fluoro-5-morpholinophenyl)-N-(4-(3-morpholino...)copy SMILEScopy InChI
Affinity DataIC50: 148nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J6JPubMedMMDB
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50224009(CHEMBL250409 | N-(tert-butyl)-4-[5-(pyridin-2-ylam...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of JNK3 by HTRF assayMore data for this Ligand-Target Pair
TargetIsoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM32460(piperazine amide, 4g)copy SMILEScopy InChI
Affinity DataIC50: 160nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM92524(Aminopyrazole inhibitor, 3576)copy SMILEScopy InChI
Affinity DataIC50: 170nMpH: 7.0 T: 2°CAssay Description:Homogeneous time-resolved fluorescence assay is an enzyme inhibition studies that were performed in 384-well polystyrene homogeneous time-resolved fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ867TPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32469(piperazine amide, 4p)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32461(piperazine amide, 4h)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetIsoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM32469(piperazine amide, 4p)copy SMILEScopy InChI
Affinity DataIC50: 200nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50224016(4-(5-(pyridin-2-ylamino)quinolin-3-yl)benzenesulfo...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of JNK3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36KXPubMed
TargetIsoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM32490(aryl piperidine, 9f)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50224002(CHEMBL250199 | N-(methylsulfonyl)-N-[4-(2,7-phenan...)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of JNK3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36KXPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32489(aryl piperidine, 9e)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32490(aryl piperidine, 9f)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32458(piperazine amide, 4e | piperazine amide, 6a)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMedMMDB
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50224008(4-(5-(5-chloropyridin-2-ylamino)quinolin-3-yl)benz...)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of JNK3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36KXPubMed
TargetIsoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402](Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM32462(piperazine amide, 4i)copy SMILEScopy InChI
Affinity DataIC50: 250nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM50224007(CHEMBL430014 | N-tert-butyl-4-(5-(5-chloropyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of JNK3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36KXPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32492(aryl piperidine, 9h)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
and Translational Research Institute

Curated by ChEMBL
LigandPNGBDBM32462(piperazine amide, 4i)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N67PubMed
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