Compile Data Set for Download or QSAR
Found 78 with Last Name = 'klint' and Initial = 'j'
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506203(CHEMBL4452312)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506156(CHEMBL4471140)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506173(CHEMBL4589444)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506179(CHEMBL4579583)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506184(CHEMBL4447043)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506180(CHEMBL4556573)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506187(CHEMBL4522504)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506201(CHEMBL4516176)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506178(CHEMBL4555657)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506183(CHEMBL4521017)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506172(CHEMBL4563994)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506185(CHEMBL4438327)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506191(CHEMBL4439570)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506169(CHEMBL4535761)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506162(CHEMBL4463320)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506157(CHEMBL4517831)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506198(CHEMBL4539658)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506166(CHEMBL4474747)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506204(CHEMBL4443234)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM393615(US09969700, 173)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human P2X4 receptor expressed in HEK cells assessed as reduction in ATP induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM393615(US09969700, 173)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506195(CHEMBL4438981)copy SMILEScopy InChI
Affinity DataIC50: 67nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506163(CHEMBL4561582)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506154(CHEMBL4516450)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506177(CHEMBL4452251)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506175(CHEMBL4519162)copy SMILEScopy InChI
Affinity DataIC50: 88nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506186(CHEMBL4449416)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506164(CHEMBL4579675)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506160(CHEMBL4513970)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human P2X4 receptor expressed in HEK cells assessed as reduction in ATP induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506205(CHEMBL4469574)copy SMILEScopy InChI
Affinity DataIC50: 111nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Mus musculus)
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)copy SMILEScopy InChI
Affinity DataIC50: 112nMAssay Description:Antagonist activity at mouse P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506182(CHEMBL4593104)copy SMILEScopy InChI
Affinity DataIC50: 134nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506174(CHEMBL4442297)copy SMILEScopy InChI
Affinity DataIC50: 139nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506188(CHEMBL4451946)copy SMILEScopy InChI
Affinity DataIC50: 163nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506200(CHEMBL4443857)copy SMILEScopy InChI
Affinity DataIC50: 173nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506171(CHEMBL4462109)copy SMILEScopy InChI
Affinity DataIC50: 185nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506197(CHEMBL4541425)copy SMILEScopy InChI
Affinity DataIC50: 193nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)copy SMILEScopy InChI
Affinity DataIC50: 211nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(RAT)
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)copy SMILEScopy InChI
Affinity DataIC50: 233nMAssay Description:Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506155(CHEMBL4577125)copy SMILEScopy InChI
Affinity DataIC50: 242nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506199(CHEMBL4450002)copy SMILEScopy InChI
Affinity DataIC50: 258nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506194(CHEMBL4462656)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506202(CHEMBL4450779)copy SMILEScopy InChI
Affinity DataIC50: 269nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506206(CHEMBL4451276)copy SMILEScopy InChI
Affinity DataIC50: 317nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of inhibition of ATP-evoked current at -90 mV hold...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506153(CHEMBL4444721)copy SMILEScopy InChI
Affinity DataIC50: 345nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506167(CHEMBL4539332)copy SMILEScopy InChI
Affinity DataIC50: 376nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506161(CHEMBL4464823)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50506168(CHEMBL4533763)copy SMILEScopy InChI
Affinity DataIC50: 441nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M048RWPubMed
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