TargetAromatase(Homo sapiens (Human))
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
CNR-IOM-Democritos c/o International School for Advanced Studies (SISSA)
Curated by ChEMBL
Affinity DataIC50: 9.53E+4nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: >8.00E+4nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.60E+5nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+4nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 800nMAssay Description:Binding affinity to 6His-tagged HMGB1 BoxA (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+4nMAssay Description:Binding affinity to 6His-tagged HMGB1 BoxB (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.60E+6nMAssay Description:Binding affinity to full-length N-terminal 6His-tagged HMGB1 (unknown origin) by NMR spectraMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+5nMAssay Description:Binding affinity to full-length N-terminal 6His-tagged HMGB1 (unknown origin) by NMR spectraMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+4nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 800nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 9.00E+5nMAssay Description:Binding affinity to full-length N-terminal 6His-tagged HMGB1 (unknown origin) by NMR spectraMore data for this Ligand-Target Pair
Affinity DataKd: 2.62E+4nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 5.80E+3nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 8.60E+3nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 800nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair
Affinity DataKd: 9.90E+3nMAssay Description:Binding affinity to 6His-tagged HMGB1 (unknown origin) incubated for 15 mins by MST analysisMore data for this Ligand-Target Pair