Compile Data Set for Download or QSAR
Found 319 with Last Name = 'tabor' and Initial = 'j'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315949((S)-N-(4-aminobutyl)-N-(2-(1-phenylethylamino)pyri...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50306491(2-(6-chloro-5-((2R,5S)-4-(1-(4-fluorophenyl)ethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52CFPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50266947(2-(6-chloro-5-((2R,5S)-4-(4-fluorobenzyl)-2,5-dime...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50306493(2-(5-((2R,5S)-4-benzhydryl-2,5-dimethylpiperazine-...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52CFPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50309525(2-(5-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-6-m...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38SP4PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315959(CHEMBL1091614 | N-(4-aminobutyl)-N-(2-(4-hydroxycy...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1VTTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315931((S)-N-ethyl-3-methyl-N-(2-(1-phenylethylamino)pyri...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mi...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315917((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315958(CHEMBL1089655 | N-(4-aminobutyl)-N-(2-(isopropylam...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50309524(2-(6-chloro-5-(4-(4-fluorobenzyl)piperidine-1-carb...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38SP4PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50570570(CHEMBL4874266)copy SMILES
Affinity DataIC50: 20nMAssay Description:Inhibition of human BuchE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1VTTPubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1VTTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315951(CHEMBL1093834 | N-(2-(isopropylamino)pyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50306492(2-(5-((2R,5S)-4-(bis(4-fluorophenyl)methyl)-2,5-di...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52CFPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315960((S)-N-(4-aminobutyl)-N-(2-(1-methoxypropan-2-ylami...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315938((S)-N-ethyl-2-fluoro-5-methyl-N-(2-(1-phenylethyla...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50306494(2-(6-chloro-5-((2R,5S)-4-(2,3-dihydro-1H-inden-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52CFPubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of human BuchE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by E...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315937((S)-N-ethyl-4-fluoro-3-methyl-N-(2-(1-phenylethyla...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315922((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetBeta-secretase 1(Homo sapiens (Human))TBA
LigandPNGBDBM16034(1-N-[(2S,3R)-4-(cyclopropylamino)-3-hydroxy-1-phen...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant human BACE1 expressed in baculovirus expression system using Rh-EVNLDAEFK-quencher as substrate incubated for 60 mins by FR...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50306496(2-(6-chloro-5-((2R,5S)-4-(1-cyano-1-(4-fluoropheny...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52CFPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50306497(2-(6-chloro-5-((2R,5S)-4-(7-chloro-1H-indazol-3-yl...)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52CFPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315943((S)-N-(2-(1-phenylethylamino)pyrimidin-4-yl)-N-(pi...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50309531(2-(5-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-6-m...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38SP4PubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM50570570(CHEMBL4874266)copy SMILES
Affinity DataIC50: 60nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1VTTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315916((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315936((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315934((S)-N,3-diethyl-N-(2-(1-phenylethylamino)pyrimidin...)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315920((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315919((S)-N-(3-(methylsulfonyl)propyl)-N-(2-(1-phenyleth...)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetCholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50570571(CHEMBL4851264)copy SMILES
Affinity DataIC50: 80nMAssay Description:Inhibition of human BuchE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1VTTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315933((S)-N-ethyl-2,3-dimethyl-N-(2-(1-phenylethylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315929((S)-3-chloro-N-ethyl-N-(2-(1-phenylethylamino)pyri...)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315921((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50309529(2-(3-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-2-m...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38SP4PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315932((S)-N-ethyl-3,4-dimethyl-N-(2-(1-phenylethylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315950((S)-N-(4-hydroxybutyl)-N-(2-(1-phenylethylamino)py...)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
Scios inc

Curated by ChEMBL
LigandPNGBDBM50266947(2-(6-chloro-5-((2R,5S)-4-(4-fluorobenzyl)-2,5-dime...)copy SMILEScopy InChI
Affinity DataIC50: 98nMAssay Description:Inhibition of p38betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52CFPubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM50570604(CHEMBL4855794)copy SMILES
Affinity DataIC50: 100nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1VTTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50309528(2-(6-chloro-5-(4-(4-fluorobenzyl)piperidine-1-carb...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38SP4PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315935((S)-3-cyclopropyl-N-ethyl-N-(2-(1-phenylethylamino...)copy SMILEScopy InChI
Affinity DataIC50: 104nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM50570589(CHEMBL4870994)copy SMILES
Affinity DataIC50: 110nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1VTTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315925((S)-N-ethyl-1-methyl-N-(2-(1-phenylethylamino)pyri...)copy SMILEScopy InChI
Affinity DataIC50: 154nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315942((S)-N-(2-(1-phenylethylamino)pyrimidin-4-yl)-N-((t...)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315918((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 164nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios Inc.

Curated by ChEMBL
LigandPNGBDBM50315940((S)-N-(cyclopropylmethyl)-N-(2-(1-phenylethylamino...)copy SMILEScopy InChI
Affinity DataIC50: 165nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7GS3PubMed
TargetCholinesterase(Equus caballus (Horse))TBA
LigandPNGBDBM50570598(CHEMBL4851448)copy SMILES
Affinity DataIC50: 170nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1VTTPubMed
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