Compile Data Set for Download or QSAR
Found 399 with Last Name = 'zhong' and Initial = 'j'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50398789(CHEMBL2180073)copy SMILEScopy InChI
Affinity DataKi:  293nMAssay Description:Inhibition of human DATMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VHKPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50398807(CHEMBL2180074)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human DATMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VHKPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50398804(CHEMBL2177497)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DATMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VHKPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50398800(CHEMBL2180069)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DATMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VHKPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553656(CHEMBL4744130)copy SMILES
Affinity DataIC50: 0.0150nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50533653(CHEMBL4519741)copy SMILEScopy InChI
Affinity DataIC50: 0.0380nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553658(CHEMBL4790915)copy SMILES
Affinity DataIC50: 0.0720nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553655(CHEMBL4749639)copy SMILES
Affinity DataIC50: 0.292nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565570(CHEMBL4798376)copy SMILES
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565559(CHEMBL4792017)copy SMILES
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565572(CHEMBL4800688)copy SMILES
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565556(CHEMBL4787929)copy SMILES
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565569(CHEMBL4780069)copy SMILES
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565571(CHEMBL4790038)copy SMILES
Affinity DataIC50: 0.577nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553660(CHEMBL4761091)copy SMILES
Affinity DataIC50: 1.20nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50533653(CHEMBL4519741)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human partial length FLT3 ITD mutant expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565558(CHEMBL4783888)copy SMILES
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565583(CHEMBL4780169)copy SMILES
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553661(CHEMBL4781811)copy SMILES
Affinity DataIC50: 1.5nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565555(CHEMBL4795375)copy SMILES
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565586(CHEMBL4799529)copy SMILES
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50533659(CHEMBL4444648)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FLT3 (564 to end residues) expressed by baculovirus in Sf21 insect cells measured after 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z76SQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565585(CHEMBL4776291)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50402023(BI 6727 | VOLASERTIB)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565577(CHEMBL4784741)copy SMILES
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553674(CHEMBL4763034)copy SMILES
Affinity DataIC50: 3.10nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553664(CHEMBL4765203)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565573(CHEMBL4785567)copy SMILES
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565582(CHEMBL4790028)copy SMILES
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553658(CHEMBL4790915)copy SMILES
Affinity DataIC50: 3.5nMAssay Description:Inhibition of FLT3 ITD/D835Y double mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565564(CHEMBL4784781)copy SMILES
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565576(CHEMBL4779654)copy SMILES
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565581(CHEMBL4800085)copy SMILES
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565557(CHEMBL4800017)copy SMILES
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565574(CHEMBL4783122)copy SMILES
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565552(CHEMBL4787496)copy SMILES
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553665(CHEMBL4763828)copy SMILES
Affinity DataIC50: 4.70nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565584(CHEMBL4778470)copy SMILES
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553672(CHEMBL4791482)copy SMILES
Affinity DataIC50: 4.90nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565575(CHEMBL4778422)copy SMILES
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565565(CHEMBL4796797)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50533653(CHEMBL4519741)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FLT3 (564 to end residues) expressed by baculovirus in Sf21 insect cells measured after 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z76SQPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553664(CHEMBL4765203)copy SMILES
Affinity DataIC50: 5.10nMAssay Description:Inhibition of FLT3 ITD/D835Y double mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565561(CHEMBL4799183)copy SMILES
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553662(CHEMBL4795857)copy SMILES
Affinity DataIC50: 5.20nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553675(CHEMBL4750430)copy SMILES
Affinity DataIC50: 5.20nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50565562(CHEMBL4790807)copy SMILES
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0KWCPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553665(CHEMBL4763828)copy SMILES
Affinity DataIC50: 5.40nMAssay Description:Inhibition of FLT3 ITD/D835Y double mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50553671(CHEMBL4749484)copy SMILES
Affinity DataIC50: 5.80nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MQ1PubMed
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