TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]-AB MECA displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]-AB MECA displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]NECA from Adenosine A2A receptor in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity at Adenosine A2A receptor in rat striatal membrane by [3H]ZM-241385 displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Ability to displace [3H]DPCPX from Adenosine A1 receptor in rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 584nMAssay Description:Displacement of [125I]APNEA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 710nMAssay Description:Ability to displace [3H]DPCPX from Adenosine A1 receptor in rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in rat cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Leiden/Amsterdam Center for Drug Research
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:G-protein activation in human adenosine Adenosine A2A receptor expressing CHO cells using cAMP assayMore data for this Ligand-Target Pair