Compile Data Set for Download or QSAR
Found 52 with Last Name = 'kritzer' and Initial = 'ja'
LigandPNGBDBM50565476(CHEMBL4780117)copy SMILES
Affinity DataIC50: 6.5nMAssay Description:Inhibition of recombinant human 10His-tagged eIF4E expressed in Escherichia coli BL21 (DE3) cells by catalytic enzyme-linked click chemistry assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W8FPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
LigandPNGBDBM50565475(CHEMBL4777401)copy SMILES
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human 10His-tagged eIF4E expressed in Escherichia coli BL21 (DE3) cells by catalytic enzyme-linked click chemistry assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W8FPubMed
LigandPNGBDBM50525088(CHEMBL4461497)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant human 10His-tagged eIF4E expressed in Escherichia coli BL21 (DE3) cells by catalytic enzyme-linked click chemistry assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W8FPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)copy SMILEScopy InChI
Affinity DataIC50: 282nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
LigandPNGBDBM50559890(CHEMBL4757551)copy SMILES
Affinity DataIC50: 410nMAssay Description:Displacement of fluorescent pTyr from recombinant His6-tagged human STAT3 (codons 127-711) expressed in Escherichia coli BL21 Rosetta after 45 mins b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CTPPubMed
LigandPNGBDBM50559892(CHEMBL4748862)copy SMILES
Affinity DataIC50: 610nMAssay Description:Displacement of fluorescent pTyr from recombinant His6-tagged human STAT3 (codons 127-711) expressed in Escherichia coli BL21 Rosetta after 45 mins b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CTPPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048520(CHEMBL3360777)copy SMILES
Affinity DataIC50: 730nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048520(CHEMBL3360777)copy SMILES
Affinity DataIC50: 4.11E+3nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
LigandPNGBDBM50559891(CHEMBL4739963)copy SMILES
Affinity DataIC50: 7.10E+3nMAssay Description:Displacement of fluorescent pTyr from recombinant His6-tagged human STAT3 (codons 127-711) expressed in Escherichia coli BL21 Rosetta after 45 mins b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CTPPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048519(CHEMBL3360776)copy SMILES
Affinity DataIC50: 8.43E+3nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048498(CHEMBL3360774)copy SMILES
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048494(CHEMBL3360770)copy SMILES
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048490(Coumermycin A1)copy SMILEScopy InChI
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048494(CHEMBL3360770)copy SMILES
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048499(CHEMBL3360775)copy SMILES
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048492(CHEMBL3360767)copy SMILES
Affinity DataIC50: 1.86E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048493(CHEMBL3360769)copy SMILES
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048519(CHEMBL3360776)copy SMILES
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453873(CHEMBL4210179)copy SMILEScopy InChI
Affinity DataIC50: 2.71E+4nMAssay Description:Inhibition of fluorescence-labelled cNPF1 probe binding to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells pretrea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048490(Coumermycin A1)copy SMILEScopy InChI
Affinity DataIC50: 2.81E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048499(CHEMBL3360775)copy SMILES
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453871(CHEMBL4203846)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of fluorescence-labelled cNPF1 probe binding to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells pretrea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048497(CHEMBL3360773)copy SMILES
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048493(CHEMBL3360769)copy SMILES
Affinity DataIC50: 3.79E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048498(CHEMBL3360774)copy SMILES
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453874(CHEMBL4218026)copy SMILEScopy InChI
Affinity DataIC50: 3.89E+4nMAssay Description:Inhibition of fluorescence-labelled cNPF1 probe binding to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells pretrea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453868(CHEMBL4214569)copy SMILEScopy InChI
Affinity DataIC50: 5.55E+4nMAssay Description:Inhibition of fluorescence-labelled cNPF1 probe binding to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells pretrea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453867(CHEMBL4205818)copy SMILEScopy InChI
Affinity DataIC50: 6.28E+4nMAssay Description:Inhibition of fluorescence-labelled cNPF1 probe binding to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells pretrea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048496(CHEMBL3360772)copy SMILES
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453869(CHEMBL4215110)copy SMILEScopy InChI
Affinity DataIC50: 6.88E+4nMAssay Description:Inhibition of fluorescence-labelled cNPF1 probe binding to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells pretrea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453866(CHEMBL4210684)copy SMILEScopy InChI
Affinity DataIC50: 7.65E+4nMAssay Description:Inhibition of fluorescence-labelled cNPF1 probe binding to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells pretrea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453872(CHEMBL4209370)copy SMILEScopy InChI
Affinity DataIC50: 8.81E+4nMAssay Description:Inhibition of fluorescence-labelled cNPF1 probe binding to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells pretrea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048492(CHEMBL3360767)copy SMILES
Affinity DataIC50: 9.45E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetEpidermal growth factor receptor substrate 15(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453870(CHEMBL4215523)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to GST-fused Eps15 EH2 domain (unknown origin) expressed in Escherichia coli BL21 cells under high salt condition by fluorescence po...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048495(CHEMBL3360771)copy SMILES
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048497(CHEMBL3360773)copy SMILES
Affinity DataIC50: 1.21E+5nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048496(CHEMBL3360772)copy SMILES
Affinity DataIC50: 1.37E+5nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048491(CHEMBL3360762)copy SMILES
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048495(CHEMBL3360771)copy SMILES
Affinity DataIC50: 1.68E+5nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90-beta(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50423645(Albamycin | Cathomycin | NOVOBIOCIN)copy SMILEScopy InChI
Affinity DataIC50: 2.31E+5nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048491(CHEMBL3360762)copy SMILES
Affinity DataIC50: 2.33E+5nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
TargetHeat shock protein HSP 90(Rabbit)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50423645(Albamycin | Cathomycin | NOVOBIOCIN)copy SMILEScopy InChI
Affinity DataIC50: 4.14E+5nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SDMPubMed
LigandPNGBDBM50565476(CHEMBL4780117)copy SMILES
Affinity DataKon:  0.00690M-1s-1Assay Description:Binding affinity to recombinant human 10His-tagged eIF4E expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by surface ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W8FPubMed
LigandPNGBDBM50525088(CHEMBL4461497)copy SMILEScopy InChI
Affinity DataKd:  17nMAssay Description:Binding affinity to recombinant human 10His-tagged eIF4E expressed in Escherichia coli BL21 (DE3) cells assessed as binding constant by surface plasm...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W8FPubMed
LigandPNGBDBM50565475(CHEMBL4777401)copy SMILES
Affinity DataKd:  7.20nMAssay Description:Binding affinity to recombinant human 10His-tagged eIF4E expressed in Escherichia coli BL21 (DE3) cells assessed as binding constant by surface plasm...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W8FPubMed
LigandPNGBDBM50565475(CHEMBL4777401)copy SMILES
Affinity DataKon:  0.00420M-1s-1Assay Description:Binding affinity to recombinant human 10His-tagged eIF4E expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by surface ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W8FPubMed
LigandPNGBDBM50525088(CHEMBL4461497)copy SMILEScopy InChI
Affinity DataKon:  0.0110M-1s-1Assay Description:Binding affinity to recombinant human 10His-tagged eIF4E expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by surface ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W8FPubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453870(CHEMBL4215523)copy SMILEScopy InChI
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells measured after 1 hr in presence of 15 mM NaCl ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
TargetEH domain-containing protein 1(Human)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50453870(CHEMBL4215523)copy SMILEScopy InChI
Affinity DataKd:  1.51E+4nMAssay Description:Binding affinity to GST-fused EHD1 EH domain (unknown origin) expressed in Escherichia coli BL21 cells measured after 1 hr in presence of 150 mM NaCl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN76G0PubMed
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