Compile Data Set for Download or QSAR
Found 39 with Last Name = 'wisniewski' and Initial = 'ja'
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014089(CHEMBL1236726)copy SMILEScopy InChI
Affinity DataKi:  109nMAssay Description:Displacement of fluorescent P4 peptide from recombinant human MDM2 (18 to 125) expressed in Escherichia coli BL21(DE3) RIL expression system after 30...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7C05PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014093(CHEMBL3260848)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Binding affinity to MDM2 (unknown origin) assessed as inhibition of interaction with p53More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7C05PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014092(CHEMBL3259830 | US9187441, 9l)copy SMILEScopy InChI
Affinity DataKi:  400nMAssay Description:Displacement of fluorescent P4 peptide from MDM2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014094(CHEMBL3260849)copy SMILEScopy InChI
Affinity DataKi:  600nMAssay Description:Binding affinity to MDM2 (unknown origin) assessed as inhibition of interaction with p53More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50436047(CHEMBL1233798)copy SMILEScopy InChI
Affinity DataKi:  916nMAssay Description:Displacement of fluorescent P4 peptide from recombinant human MDM2 (18 to 125) expressed in Escherichia coli BL21(DE3) RIL expression system after 30...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014090(CHEMBL3260846)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of fluorescent P4 peptide from recombinant human MDM2 (18 to 125) expressed in Escherichia coli BL21(DE3) RIL expression system after 30...More data for this Ligand-Target Pair
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014098(CHEMBL3260852)copy SMILEScopy InChI
Affinity DataKi:  1.35E+3nMAssay Description:Inhibition of beta-catenin/T cell factor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7C05PubMed
TargetCatenin beta-1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014148(CHEMBL3260853)copy SMILEScopy InChI
Affinity DataKi:  1.36E+3nMAssay Description:Competitive binding affinity to human beta-catenin (142 to 686) assessed as inhibition of C-terminally fluorescein-labeled Tcf4 interaction after 3 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7C05PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014091(CHEMBL3260847)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of fluorescent P4 peptide from MDM2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7C05PubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501088(CHEMBL3819630)copy SMILEScopy InChI
Affinity DataKi:  2.10E+3nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetCatenin beta-1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014132(CHEMBL2323032)copy SMILEScopy InChI
Affinity DataKi:  3.14E+3nMAssay Description:Competitive binding affinity to human beta-catenin (142 to 686) assessed as inhibition of C-terminally fluorescein-labeled Tcf4 interaction after 3 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7C05PubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501080(CHEMBL3819506)copy SMILEScopy InChI
Affinity DataKi:  5.20E+3nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50371232(CARNOSIC ACID)copy SMILEScopy InChI
Affinity DataKi:  5.30E+3nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501081(CHEMBL3819020)copy SMILEScopy InChI
Affinity DataKi:  1.60E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501086(CHEMBL3818707)copy SMILEScopy InChI
Affinity DataKi:  1.90E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501079(CHEMBL3819288)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501083(CHEMBL3819165)copy SMILEScopy InChI
Affinity DataKi:  2.50E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501078(CHEMBL3818097)copy SMILEScopy InChI
Affinity DataKi:  3.50E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501092(CHEMBL3819088)copy SMILEScopy InChI
Affinity DataKi:  3.70E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501093(CHEMBL3818263)copy SMILEScopy InChI
Affinity DataKi:  4.50E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501090(CHEMBL3819332)copy SMILEScopy InChI
Affinity DataKi:  4.80E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501082(CHEMBL3818667)copy SMILEScopy InChI
Affinity DataKi:  5.30E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501085(CHEMBL3818058)copy SMILEScopy InChI
Affinity DataKi:  5.50E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501091(CHEMBL3819368)copy SMILEScopy InChI
Affinity DataKi:  5.70E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501077(CHEMBL3818956)copy SMILEScopy InChI
Affinity DataKi:  6.70E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501084(CHEMBL3818280)copy SMILEScopy InChI
Affinity DataKi:  6.90E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501097(CHEMBL3818207)copy SMILEScopy InChI
Affinity DataKi:  7.00E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501094(CHEMBL3817935)copy SMILEScopy InChI
Affinity DataKi:  7.60E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501089(CHEMBL3818949)copy SMILEScopy InChI
Affinity DataKi:  8.20E+4nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501087(CHEMBL3818840)copy SMILEScopy InChI
Affinity DataKi:  1.30E+5nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetCatenin beta-1/B-cell CLL/lymphoma 9 protein(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501076(CHEMBL3819443)copy SMILEScopy InChI
Affinity DataKi:  1.70E+5nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501096(CHEMBL3818029)copy SMILEScopy InChI
Affinity DataKi:  4.90E+5nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501095(CHEMBL3818748)copy SMILEScopy InChI
Affinity DataKi: >5.00E+5nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetElongin-C(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014097(CHEMBL3260851)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Displacement of FAM-DEALAHyp-YIPD from VHL/elongins-B/elonginC (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetElongin-C(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50446138(CHEMBL3108881)copy SMILEScopy InChI
Affinity DataIC50: 4.10E+3nMAssay Description:Displacement of FAM-DEALAHyp-YIPD from 6xHis-tagged VHL (1 to 213)/elongins-B/elonginC (unknown origin) expressed in Escherichia coli BL21 after 1 mi...More data for this Ligand-Target Pair
TargetB-cell CLL/lymphoma 9 protein(Homo sapiens)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50501080(CHEMBL3819506)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Competitive inhibition of wild type beta-catenin (unknown origin) expressed in Escherichia coli BL21 DE3 interaction with N-terminally biotinylated h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43X4JPubMed
TargetElongin-B/Elongin-C/von Hippel-Lindau disease tumor suppressor(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014095(CHEMBL3260850)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+5nMAssay Description:Displacement of FAM-DEALAHyp-YIPD from 6xHis-tagged VHL (1 to 213)/elongins-B/elonginC (unknown origin) expressed in Escherichia coli BL21 after 1 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7C05PubMed
TargetInterferon alpha/beta receptor 1(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014088(CHEMBL1617534 | DNDI1417107)copy SMILEScopy InChI
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to IFNAR (unknown origin) assessed as inhibition of interaction with IFN-alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7C05PubMed
TargetElongin-C(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50446134(CHEMBL3108877)copy SMILEScopy InChI
Affinity DataKd:  1.00E+7nMAssay Description:Displacement of FAM-DEALAHyp-YIPD from VHL/elongins-B/elonginC (unknown origin) by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair