Compile Data Set for Download or QSAR
Found 35 with Last Name = 'chabala' and Initial = 'jc'
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))copy SMILEScopy InChI
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280339((S)-2-[4-(2-Benzenesulfonyl-ethoxy)-3-methoxy-5-(p...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Compound was evaluated for inhibition of binding of [3H]-C18 PAF to human platelet membrane Platelet activating factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X588Z
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002827(1-{3-(3-Hydroxy-propoxy)-2-propoxy-5-[(2S,5S)-5-(3...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002828(1-{3-(3-Morpholin-4-yl-propoxy)-2-propoxy-5-[(2S,5...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002824((S)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-tri...)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002827(1-{3-(3-Hydroxy-propoxy)-2-propoxy-5-[(2S,5S)-5-(3...)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002826(1-{3-(3-Imidazol-1-yl-propoxy)-2-propoxy-5-[(2S,5S...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002825((R)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-tri...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002824((S)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-tri...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002825((R)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-tri...)copy SMILEScopy InChI
Affinity DataKi:  3.72nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM82381(L-659,989, (-))copy SMILEScopy InChI
Affinity DataKi:  5.48nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:In vitro inhibition of [3H]-C18 PAF binding to human platelet membrane Platelet activating factor receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X588Z
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to PMN membrane receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM81972((S)-(+)-ALPHA-METHYL-1H-IMIDAZOLE-4-ETHANAMINE DIH...)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  12.2nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM81972((S)-(+)-ALPHA-METHYL-1H-IMIDAZOLE-4-ETHANAMINE DIH...)copy SMILEScopy InChI
Affinity DataKi:  14.3nMAssay Description:In vitro inhibition of [3H]-C18 PAF binding to human platelet membrane Platelet activating factor receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X588Z
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  14.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)copy SMILEScopy InChI
Affinity DataKi:  79.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366241(CHEMBL297624 | L-652731)copy SMILEScopy InChI
Affinity DataKi:  103nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366241(CHEMBL297624 | L-652731)copy SMILEScopy InChI
Affinity DataKi:  103nMAssay Description:Inhibitory concentration required to inhibit PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002822((-)-trans 42s,5S)-2-[3-[(2-Oxopropyl)sulfony1]-4-n...)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  152nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002822((-)-trans 42s,5S)-2-[3-[(2-Oxopropyl)sulfony1]-4-n...)copy SMILEScopy InChI
Affinity DataKi:  174nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  205nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002830((2R,3R,4R,5S)-2,5-Bis-(3,4-dimethoxy-phenyl)-3,4-d...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  1.11E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280339((S)-2-[4-(2-Benzenesulfonyl-ethoxy)-3-methoxy-5-(p...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Compound was evaluated for inhibitory activity of binding of [3H]-C18 PAF to human platelet membrane Platelet activating factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X588Z
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50001747((+)-Kadsurenone | (Kadsurenone)5-Allyl-2-(3,4-dime...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibitory concentration required to inhibit PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50002830((2R,3R,4R,5S)-2,5-Bis-(3,4-dimethoxy-phenyl)-3,4-d...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration required to inhibit PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP