Compile Data Set for Download or QSAR
Found 290 with Last Name = 'mckelvie' and Initial = 'jc'
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107257(CHEMBL3600785)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107256(CHEMBL3600784)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107248(CHEMBL3600781)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107243(CHEMBL3600779)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107254(CHEMBL3600782)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107255(CHEMBL3600783)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107263(CHEMBL3600687)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107260(CHEMBL3600684)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50107273(CHEMBL3600699)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of PI3Kgamma (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107258(CHEMBL3600683)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107238(CHEMBL3600776)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50107273(CHEMBL3600699)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of PI3Kbeta (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plus...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50107273(CHEMBL3600699)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of PI3Kalpha (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107257(CHEMBL3600785)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50107272(CHEMBL3600698)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of PI3Kgamma (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107261(CHEMBL3600685)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107242(CHEMBL3600778)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50106970(CHEMBL3600767)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107269(CHEMBL3600694)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107242(CHEMBL3600778)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107241(CHEMBL3600777)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107270(CHEMBL3600695)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107254(CHEMBL3600782)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50107273(CHEMBL3600699)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of PI3Kdelta (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107248(CHEMBL3600781)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50333219(6-(6-methoxypyridin-3-yl)benzo[d]thiazol-2-amine |...)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of PI3Kgamma (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107273(CHEMBL3600699)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107277(CHEMBL97245)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107269(CHEMBL3600694)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50107272(CHEMBL3600698)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of PI3Kalpha (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107241(CHEMBL3600777)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107266(CHEMBL3600691)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50106926(CHEMBL3600701)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50106970(CHEMBL3600767)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107260(CHEMBL3600684)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107258(CHEMBL3600683)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50333219(6-(6-methoxypyridin-3-yl)benzo[d]thiazol-2-amine |...)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107236(CHEMBL3600775)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107265(CHEMBL3600689)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107264(CHEMBL3600688)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107256(CHEMBL3600784)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107244(CHEMBL3600780)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of N-terminal FLAG-tagged human full length recombinant PI4K3alpha using D-myo-phosphatidylinositol substrate and ATP incubated for 45 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107275(CHEMBL3600690)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50333219(6-(6-methoxypyridin-3-yl)benzo[d]thiazol-2-amine |...)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Inhibition of PI3Kalpha (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107238(CHEMBL3600776)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
LigandPNGBDBM50333219(6-(6-methoxypyridin-3-yl)benzo[d]thiazol-2-amine |...)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Inhibition of PI3Kdelta (unknown origin) pre-incubated for 20 mins before phosphatidylinositol 4, 5-bisphosphate substrate addition by kinase-glo plu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)copy SMILEScopy InChI
Affinity DataIC50: 941nMAssay Description:Inhibition of human Dnmt1 using oligonucleotide 2 as substrate after 5000 sec by micro plate reader based real-time break-light assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50333221(6-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107012(CHEMBL3600769)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50107272(CHEMBL3600698)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal GST-tagged human full length recombinant PI4K3beta expressed in Sf9 cells using D-myo-phosphatidylinositol substrate and ATP...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9DKRPubMed
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