Compile Data Set for Download or QSAR
Found 88 with Last Name = 'tomassini' and Initial = 'je'
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144942(2'-C-Me-guanosine | 2'-C-methyl-guanosine | 2'-C-m...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385528(CHEMBL2040586)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of Influenza replicationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ09B6PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385503(CHEMBL2040554)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ09B6PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125801(4-[1-Benzyl-4-(4-chloro-benzyl)-piperidin-4-yl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of Influenza replicationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ09B6PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125801(4-[1-Benzyl-4-(4-chloro-benzyl)-piperidin-4-yl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ09B6PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385528(CHEMBL2040586)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ09B6PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144937(2-Amino-9-((2R,3R,5S)-3-hydroxy-5-hydroxymethyl-te...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385503(CHEMBL2040554)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of Influenza replicationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ09B6PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385531(CHEMBL2040602)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125833(3-(4-Fluoro-benzylidene)-1-hydroxy-5-isobutyl-3H-p...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385529(CHEMBL2040587)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ09B6PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385532(CHEMBL2040603)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385529(CHEMBL2040587)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Influenza replicationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ09B6PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144947(2-Amino-9-((2R,3R,4R,5R)-4-hydroxy-5-hydroxymethyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144938(2-Amino-9-((2R,3S,4S,5R)-4-fluoro-3-hydroxy-5-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144948((2R,3R,4R,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144949((2R,3R,4R,5R)-2-(2,6-diamino-9H-purin-9-yl)-5-(hyd...)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385534(CHEMBL2040605)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385535(CHEMBL2040606)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144934((2R,3R,4R,5R)-2-(6-hydroxy-9H-purin-9-yl)-5-(hydro...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385530(CHEMBL2040601)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125822(1-Hydroxy-5-isobutyl-3-isobutylidene-3H-pyrazine-2...)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385536(CHEMBL2040608)copy SMILEScopy InChI
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385533(CHEMBL2040604)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409930(CHEMBL2021379)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144950(3'-deoxyadenosine | 9-(beta-D-3'-Deoxyribofuranosy...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144933((2R,3S,4S,5R)-4-Fluoro-5-hydroxymethyl-2-(6-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144939((2R,3R,4R,5R)-2-(2-amino-9H-purin-9-yl)-5-(hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144945((2R,3R,4R,5R)-2-Hydroxymethyl-4-methoxy-5-(6-methy...)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144940((2R,3S,4R,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144936(CHEMBL1090 | VIDARABINE | adenine arabinoside)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144941((2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-2-(hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408410(CHEMBL480143)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144932((2R,3R,4R,5R)-4-Fluoro-2-hydroxymethyl-5-(6-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144935((2R,3R,4R,5R)-2-(6-amino-9H-purin-9-yl)-3-ethyl-5-...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50422565(CHEMBL2311161)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2BQ3PubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385561(CHEMBL2040639)copy SMILEScopy InChI
Affinity DataIC50: 8.50E+4nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385545(CHEMBL2040618)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385550(CHEMBL2040625)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385557(CHEMBL2040634)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385537(CHEMBL2040609)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385538(CHEMBL2040610)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385539(CHEMBL2040611)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385540(CHEMBL2040612)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385541(CHEMBL2040613)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385542(CHEMBL2040614)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385543(CHEMBL2040616)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385544(CHEMBL2040617)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385546(CHEMBL2040620)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385547(CHEMBL2040621)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q298882DPubMed
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