Compile Data Set for Download or QSAR
Found 110 with Last Name = 'douglass' and Initial = 'jg'
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371580(CHEMBL1162175)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371581(CHEMBL1162179)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374555(REGRELOR DISODIUM)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371580(CHEMBL1162175)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371582(CHEMBL1162182)copy SMILEScopy InChI
Affinity DataIC50: 36.2nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374558(CHEMBL255350)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371583(CHEMBL1162184)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371589(CHEMBL1162196)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371594(CHEMBL1162161)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371584(CHEMBL1162185)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371585(CHEMBL1162188)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374572(CHEMBL403010)copy SMILEScopy InChI
Affinity DataIC50: 201nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371578(CHEMBL1162172)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371577(CHEMBL1162173)copy SMILEScopy InChI
Affinity DataIC50: 211nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371579(CHEMBL1162171)copy SMILEScopy InChI
Affinity DataIC50: 237nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374559(CHEMBL255349)copy SMILEScopy InChI
Affinity DataIC50: 243nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371576(CHEMBL1162164)copy SMILEScopy InChI
Affinity DataIC50: 288nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374571(CHEMBL272113)copy SMILEScopy InChI
Affinity DataIC50: 495nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374566(CHEMBL272975)copy SMILEScopy InChI
Affinity DataIC50: 513nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371593(CHEMBL1162159)copy SMILEScopy InChI
Affinity DataIC50: 522nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374568(CHEMBL401780)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374557(CHEMBL267283)copy SMILEScopy InChI
Affinity DataIC50: 616nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374560(CHEMBL256251)copy SMILEScopy InChI
Affinity DataIC50: 663nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374574(CHEMBL265707)copy SMILEScopy InChI
Affinity DataIC50: 1.27E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374556(CHEMBL412171)copy SMILEScopy InChI
Affinity DataIC50: 1.31E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371603(CHEMBL1162165)copy SMILEScopy InChI
Affinity DataIC50: 1.82E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374565(CHEMBL403011)copy SMILEScopy InChI
Affinity DataIC50: 2.23E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374561(CHEMBL427723)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374564(CHEMBL255553)copy SMILEScopy InChI
Affinity DataIC50: 2.49E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374567(CHEMBL269934)copy SMILEScopy InChI
Affinity DataIC50: 2.55E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374569(CHEMBL271643)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374575(CHEMBL403928)copy SMILEScopy InChI
Affinity DataIC50: 2.95E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371589(CHEMBL1162196)copy SMILEScopy InChI
Affinity DataIC50: 3.06E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371588(CHEMBL1162195)copy SMILEScopy InChI
Affinity DataIC50: 3.11E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371573(CHEMBL1162158)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371573(CHEMBL1162158)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374562(CHEMBL402401)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374570(CHEMBL402592)copy SMILEScopy InChI
Affinity DataIC50: 4.33E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371599(CHEMBL1162169)copy SMILEScopy InChI
Affinity DataIC50: 4.63E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374573(CHEMBL260602)copy SMILEScopy InChI
Affinity DataIC50: 4.73E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374576(CHEMBL402800)copy SMILEScopy InChI
Affinity DataIC50: 4.86E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371598(CHEMBL1162170)copy SMILEScopy InChI
Affinity DataIC50: 6.54E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371571(CHEMBL1162181)copy SMILEScopy InChI
Affinity DataIC50: 7.59E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371570(CHEMBL1162162)copy SMILEScopy InChI
Affinity DataIC50: 8.29E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371574(CHEMBL1162157)copy SMILEScopy InChI
Affinity DataIC50: 8.68E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371574(CHEMBL1162157)copy SMILEScopy InChI
Affinity DataIC50: 8.80E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50374563(CHEMBL257651)copy SMILEScopy InChI
Affinity DataIC50: 9.90E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM885RPubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371601(CHEMBL1162189)copy SMILEScopy InChI
Affinity DataIC50: 1.07E+4nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371596(CHEMBL1162163)copy SMILEScopy InChI
Affinity DataIC50: 1.08E+4nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371592(CHEMBL1162205)copy SMILEScopy InChI
Affinity DataIC50: 1.12E+4nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PB6PubMed
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