Compile Data Set for Download or QSAR
Found 134 with Last Name = 'andersen' and Initial = 'jh'
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557298(CHEMBL4750927)copy SMILES
Affinity DataKi:  30nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557293(CHEMBL4781637)copy SMILES
Affinity DataKi:  40nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557299(CHEMBL4799812)copy SMILES
Affinity DataKi:  170nMAssay Description:Binding affinity to syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557299(CHEMBL4799812)copy SMILES
Affinity DataKi:  190nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557296(CHEMBL4792861)copy SMILES
Affinity DataKi:  250nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557297(CHEMBL4747962)copy SMILES
Affinity DataKi:  250nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557295(CHEMBL4758599)copy SMILES
Affinity DataKi:  250nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557294(CHEMBL4749490)copy SMILES
Affinity DataKi:  250nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557287(CHEMBL4752622)copy SMILES
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557286(CHEMBL4798461)copy SMILES
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557288(CHEMBL4792781)copy SMILES
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Troms£

Curated by ChEMBL
LigandPNGBDBM50446576(CHEMBL3109481)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Noncompetitive inhibition of electric eel AChE using acetylthiocholine chloride as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49S8BPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557289(CHEMBL4740875)copy SMILES
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557290(CHEMBL4798840)copy SMILES
Affinity DataKi:  4.40E+4nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Troms£

Curated by ChEMBL
LigandPNGBDBM50446577(CHEMBL3109482)copy SMILEScopy InChI
Affinity DataKi:  9.00E+4nMAssay Description:Noncompetitive inhibition of electric eel AChE using acetylthiocholine chloride as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49S8BPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557291(CHEMBL4785814)copy SMILES
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557292(CHEMBL4779632)copy SMILES
Affinity DataKi:  1.10E+5nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSyntenin-1(Homo sapiens)TBA
LigandPNGBDBM50557285(CHEMBL4788058)copy SMILES
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CRXPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509371(CHEMBL4521241)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)copy SMILEScopy InChI
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK2 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
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