Compile Data Set for Download or QSAR
Found 186 with Last Name = 'dao' and Initial = 'jh'
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50264220(2-(1,6-diphenyl-1H-imidazo[4,5-c]pyridine-4-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PHD2 (unknown origin) by fluorescence energy transfer analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2WB7PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50251959(2-(2-(2-(4-tert-butylbenzylsulfonyl)acetamido)-3-h...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016165(CHEMBL3261516)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016166(CHEMBL3261517)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 2 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 1 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50251958(2-(2-(2-(benzylsulfonyl)acetamido)-3-hydroxy-2,3-d...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 6 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.667 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016148(CHEMBL3261500)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.012 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016161(CHEMBL3261512)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016160(CHEMBL3261511)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 9 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.333 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50251957(CHEMBL519615 | {2-[2-(Biphenyl-4-sulfonyl)-acetyli...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
LigandPNGBDBM50016167(CHEMBL3261518)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50252002(2-(2-(2-(4-tert-butylphenylsulfonyl)acetamido)-3-h...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 18 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50251908(2-(3-hydroxy-2-(2-(naphthalen-2-ylsulfonyl)acetami...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.111 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016162(CHEMBL3261513)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50251907(2-(2-(2-(4-chlorophenylsulfonyl)acetamido)-3-hydro...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.222 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.025 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016153(CHEMBL3261505)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 27 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50252001(2-(3-hydroxy-2-(2-tosylacetamido)-2,3-dihydrothiaz...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
LigandPNGBDBM50016164(CHEMBL3261515)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.037 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.074 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50264219(2-(6-chloro-1-phenyl-1H-imidazo[4,5-c]pyridine-4-c...)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of PHD2 (unknown origin) by fluorescence energy transfer analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2WB7PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50251900(2-(3-hydroxy-2-(2-(phenylsulfonyl)acetamido)-2,3-d...)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50251905(2-(2-(2-(2-chlorophenylsulfonyl)acetamido)-3-hydro...)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
TargetCasein kinase I isoform delta(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of CK1delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016163(CHEMBL3261514)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 54 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016147(CHEMBL3261499)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50251906(2-(2-(2-(3-chlorophenylsulfonyl)acetamido)-3-hydro...)copy SMILEScopy InChI
Affinity DataIC50: 98nMAssay Description:Inhibition of human PHD2 assesssed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4JM5PubMed
LigandPNGBDBM50016137(CHEMBL3261489)copy SMILEScopy InChI
Affinity DataIC50: 101nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetCasein kinase I isoform delta(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50016166(CHEMBL3261517)copy SMILEScopy InChI
Affinity DataIC50: 104nMAssay Description:Inhibition of CK1delta (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016146(CHEMBL3261498)copy SMILEScopy InChI
Affinity DataIC50: 104nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016136(CHEMBL3261488)copy SMILEScopy InChI
Affinity DataIC50: 115nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016135(CHEMBL3261245)copy SMILEScopy InChI
Affinity DataIC50: 172nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50264174(2-(1-phenyl-1H-imidazo[4,5-c]pyridine-4-carboxamid...)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of PHD2 (unknown origin) by fluorescence energy transfer analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2WB7PubMed
LigandPNGBDBM50016116(CHEMBL3261228)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.023 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016116(CHEMBL3261228)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 0.75 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
LigandPNGBDBM50016116(CHEMBL3261228)copy SMILEScopy InChI
Affinity DataIC50: 318nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin) using 1.5 uM of ATP as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
TargetEgl nine homolog 1(Human)
Amgen, Inc.

Curated by ChEMBL
LigandPNGBDBM50264175(2-(1-benzyl-1H-imidazo[4,5-c]pyridine-4-carboxamid...)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of PHD2 (unknown origin) by fluorescence energy transfer analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2WB7PubMed
LigandPNGBDBM50016116(CHEMBL3261228)copy SMILEScopy InChI
Affinity DataIC50: 323nMAssay Description:Inhibition of Cdc7/Dbf4 (unknown origin)-mediated phosphorylation of MCM2 by protein-A luminescent proximity homogenous assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62R8PubMed
Displayed 1 to 50 (of 186 total ) | Next | Last >>
Jump to: