Compile Data Set for Download or QSAR
Found 13 with Last Name = 'sakamoto' and Initial = 'ji'
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50260529(CHEMBL4077626)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of C-terminal biotin-labelled BCoR (Arg498 to 514Pro residues) binding to recombinant FLAG-tagged BCL6 BTB (5 to 129 residues) (unknown or...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SR7PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50260534(CHEMBL4066375)copy SMILEScopy InChI
Affinity DataIC50: 2.12E+5nMAssay Description:Inhibition of C-terminal biotin-labelled BCoR/wild-type BCL6 BTB domain (unknown origin) protein-protein interaction by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SR7PubMed
TargetGTPase KRas(Homo sapiens (Human))
Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited, 26-1, Muraoka-Higashi 2-chome, Fujisawa, Kanagawa 251-8555, Japan.

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)copy SMILEScopy InChI
Affinity DataKd:  35nMAssay Description:Binding affinity to human N-terminal His/AVi-tagged biotinylated GTPase KRas G12C mutant expressed in Escherichia coli BL21 (DE3) in presence of GDP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40XNFPubMed
TargetGTPase KRas(Homo sapiens (Human))
Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited, 26-1, Muraoka-Higashi 2-chome, Fujisawa, Kanagawa 251-8555, Japan.

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)copy SMILEScopy InChI
Affinity DataKd:  250nMAssay Description:Binding affinity to human N-terminal His/AVi-tagged biotinylated GTPase KRas G12C mutant expressed in Escherichia coli BL21 (DE3) in presence of GTP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40XNFPubMed
TargetGTPase KRas(Homo sapiens (Human))
Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited, 26-1, Muraoka-Higashi 2-chome, Fujisawa, Kanagawa 251-8555, Japan.

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)copy SMILEScopy InChI
Affinity DataKd:  200nMAssay Description:Binding affinity to human wild type N-terminal His/AVi-tagged biotinylated KRas expressed in Escherichia coli BL21 (DE3) in presence of GTP by SPR as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40XNFPubMed
TargetGTPase KRas(Homo sapiens (Human))
Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited, 26-1, Muraoka-Higashi 2-chome, Fujisawa, Kanagawa 251-8555, Japan.

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)copy SMILEScopy InChI
Affinity DataKd:  58nMAssay Description:Binding affinity to human wild type N-terminal His/AVi-tagged biotinylated KRas expressed in Escherichia coli BL21 (DE3) in presence of GDP by SPR as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40XNFPubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50260529(CHEMBL4077626)copy SMILEScopy InChI
Affinity DataKd:  0.570nMAssay Description:Binding affinity to biotinylated BCL6 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SR7PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50260528(CHEMBL4063725)copy SMILEScopy InChI
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to wild-type avi-tagged BCL6 BTB domain (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50239395(CHEMBL4061302)copy SMILEScopy InChI
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to recombinant RED-NHS labelled BCL6 BTB domain (1 to 129 residues) (unknown origin) after 10 mins by microscale thermophoresis meth...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SR7PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50260534(CHEMBL4066375)copy SMILEScopy InChI
Affinity DataKd:  1.29E+5nMAssay Description:Binding affinity to recombinant RED-NHS labelled BCL6 BTB domain (1 to 129 residues) (unknown origin) after 10 mins by microscale thermophoresis meth...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SR7PubMed
TargetGTPase KRas(Homo sapiens (Human))
Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited, 26-1, Muraoka-Higashi 2-chome, Fujisawa, Kanagawa 251-8555, Japan.

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)copy SMILEScopy InChI
Affinity DataKd:  11nMAssay Description:Binding affinity to human N-terminal His/AVi-tagged biotinylated GTPase KRas G12D mutant (1 to 169 residues) expressed in Escherichia coli BL21 (DE3)...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40XNFPubMed
TargetGTPase KRas(Homo sapiens (Human))
Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited, 26-1, Muraoka-Higashi 2-chome, Fujisawa, Kanagawa 251-8555, Japan.

Curated by ChEMBL
LigandPNGBDBM50242325(CHEMBL4072295)copy SMILEScopy InChI
Affinity DataKd:  200nMAssay Description:Binding affinity to human wild type N-terminal His/AVi-tagged biotinylated KRas expressed in Escherichia coli BL21 (DE3) in presence of GTP by SPR as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40XNFPubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50260527(CHEMBL4096591)copy SMILEScopy InChI
Affinity DataKd:  2.40E+4nMAssay Description:Binding affinity to wild-type avi-tagged BCL6 BTB domain (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SR7PubMed